SCHEMBL688172

SCHEMBL688172

CCOc1cccc(Cl)c1Cn1ccc(O)c(NC(=O)N[C@@H](CC(=O)O)c2ccc(C)cc2)c1=O

nearest known ligand 0.41

Predicted protein targets (top 15)

geneUniProtsupporting neighboursconfidence
MAPT P10636 1/20 0.41
CTSA P10619 8/20 0.40
KDM4E B2RXH2 3/20 0.38
ALDH1A1 P00352 3/20 0.38
MAPK1 P28482 1/20 0.38
SMN1; SMN2 Q16637 2/20 0.38
ITGB1 P05556 2/20 0.37
ITGA4 P13612 2/20 0.37
HPGD P15428 1/20 0.36
POLB P06746 2/20 0.35
MEN1 O00255 1/20 0.35
KMT2A Q03164 1/20 0.35
PKM P14618 1/20 0.35
NPSR1 Q6W5P4 1/20 0.35
RXFP1 Q9HBX9 1/20 0.35

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL687232 0.93 CTSA (0.46) CTSAKDM4EALDH1A1MAPK1POLB
SCHEMBL688530 0.92 CTSA (0.43) MAPTCTSAKDM4EALDH1A1MAPK1
SCHEMBL688247 0.90 SMN1; SMN2 (0.39) MAPTCTSAKDM4EALDH1A1SMN1; SMN2
SCHEMBL28780278 0.90 SMN1; SMN2 (0.39) MAPTCTSAKDM4EALDH1A1SMN1; SMN2
SCHEMBL687715 0.89 CTSA (0.39) MAPTCTSAKDM4EALDH1A1MAPK1
SCHEMBL27762477 0.89 SMN1; SMN2 (0.39) MAPTKDM4EALDH1A1MAPK1SMN1; SMN2
SCHEMBL688103 0.88 ALDH1A1 (0.51) MAPTCTSAKDM4EALDH1A1MAPK1
SCHEMBL7589554 0.88 ALDH1A1 (0.51) MAPTCTSAKDM4EALDH1A1MAPK1
SCHEMBL687573 0.88 SMN1; SMN2 (0.38) MAPTKDM4EALDH1A1SMN1; SMN2ITGB1
SCHEMBL687335 0.87 CTSA (0.43) CTSAPOLB

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1203766-B1 Carboxylic acid derivatives that inhibit the binding of integrins to their receptors ENCYSIVE PHARMACEUTICALS INC (US) 2012-02-29 EP disclosed
EP-1203766-A2 Carboxylic acid derivatives that inhibit the binding of integrins to their receptors TEXAS BIOTECHNOLOGY CORPORATION (US) 2002-05-08 EP disclosed