SCHEMBL6882464

SCHEMBL6882464

CC(=O)NC1CC1Sc1nc(C)cc2c1c(=O)cc(Nc1ccccc1)n2-c1ccccc1

nearest known ligand 0.36

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
PDE11A Q9HCR9 1/20 0.36
MAPT P10636 6/20 0.34
ALDH1A1 P00352 6/20 0.34
KDM4E B2RXH2 3/20 0.34
NPC1 O15118 3/20 0.34
THRB P10828 1/20 0.34
HSD17B10 Q99714 1/20 0.34
GAA P10253 4/20 0.32
CNR1 P21554 2/20 0.32
CNR2 P34972 2/20 0.32
GFER P55789 1/20 0.32
HPGD P15428 3/20 0.32
MAPK1 P28482 1/20 0.32
SMN1; SMN2 Q16637 4/20 0.32
LMNA P02545 3/20 0.32
MEN1 O00255 2/20 0.32
KMT2A Q03164 2/20 0.32
RAB9A P51151 2/20 0.32
CLK1 P49759 1/20 0.32
POLB P06746 1/20 0.32

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7046873 0.80 PDE11A (0.37) PDE11AMAPTALDH1A1KDM4ENPC1
SCHEMBL5872104 0.79 GAA (0.45) PDE11AKDM4ENPC1HSD17B10GAA
SCHEMBL5872280 0.78 ALDH1A1 (0.46) ALDH1A1KDM4EGAASMN1; SMN2LMNA
SCHEMBL8287549 0.78 PDE11A (0.39) PDE11AMAPTALDH1A1KDM4ENPC1
SCHEMBL7036674 0.77 ALDH1A1 (0.41) PDE11AMAPTALDH1A1GAAHPGD
SCHEMBL5872094 0.77 PDE11A (0.40) PDE11AMAPTALDH1A1KDM4ENPC1
SCHEMBL8286548 0.76 SMN1; SMN2 (0.50) MAPTNPC1GAAMAPK1SMN1; SMN2
SCHEMBL5871645 0.76 GAA (0.42) PDE11AMAPTALDH1A1KDM4ENPC1
SCHEMBL5871665 0.76 GAA (0.36) PDE11AKDM4EGAAGFERHPGD
SCHEMBL8287221 0.76 APLNR (0.42) PDE11AMAPTALDH1A1KDM4EGAA

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-1578781-A 1, 8-naphthyridine derivatives useful as antidiabetic agents BAYER PHARMACEUTICALS CORP (US) 2005-02-09 CN disclosed
CN-1578780-A 1, 6-naphthyridine derivatives useful as antidiabetic agents BAYER PHARMACEUTICALS CORP (US) 2005-02-09 CN disclosed
US-6677352-B1 1,6-naphthyridine derivatives and their use to treat diabetes and related disorders BAYER PHARMACEUTICALS CORPORATION 2004-01-13 US disclosed