SCHEMBL688356

SCHEMBL688356

COc1ccc(C(C)=O)cc1Cn1ccc(O)c(NC(=O)N[C@@H](CC(=O)O)c2ccc(C)cc2)c1=O

nearest known ligand 0.45

Predicted protein targets (top 7)

geneUniProtsupporting neighboursconfidence
CTSA P10619 13/20 0.45
POLB P06746 1/20 0.40
MAPK1 P28482 1/20 0.39
HTT P42858 1/20 0.39
ALDH1A1 P00352 3/20 0.39
SMN1; SMN2 Q16637 1/20 0.39
RXFP1 Q9HBX9 1/20 0.38

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL687559 0.88 ALDH1A1 (0.49) CTSAPOLBALDH1A1
SCHEMBL687449 0.85 CTSA (0.47) CTSAPOLB
SCHEMBL687335 0.83 CTSA (0.43) CTSAPOLB
SCHEMBL687896 0.82 CTSA (0.41) CTSAPOLB
SCHEMBL688035 0.82 CTSA (0.41) CTSAPOLBALDH1A1RXFP1
SCHEMBL687690 0.81 CTSA (0.44) CTSA
SCHEMBL687511 0.81 MEN1 (0.46) CTSAPOLBALDH1A1SMN1; SMN2
SCHEMBL688264 0.81 LCK (0.47) CTSAPOLBMAPK1ALDH1A1RXFP1
SCHEMBL687280 0.81 POLB (0.43) CTSAPOLB
SCHEMBL687925 0.80 CYP26A1 (0.42) CTSAPOLBALDH1A1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1203766-B1 Carboxylic acid derivatives that inhibit the binding of integrins to their receptors ENCYSIVE PHARMACEUTICALS INC (US) 2012-02-29 EP disclosed
EP-1203766-A2 Carboxylic acid derivatives that inhibit the binding of integrins to their receptors TEXAS BIOTECHNOLOGY CORPORATION (US) 2002-05-08 EP disclosed