SCHEMBL688220

SCHEMBL688220

Cc1ccc([C@H](CC(=O)O)NC(=O)Nc2c(O)c(C)cn(Cc3c(C)cccc3Cl)c2=O)cc1C

nearest known ligand 0.38

Predicted protein targets (top 15)

geneUniProtsupporting neighboursconfidence
SLC22A12 Q96S37 3/20 0.36
CYP26A1 O43174 2/20 0.36
KDM4E B2RXH2 3/20 0.36
ALDH1A1 P00352 3/20 0.36
CYP3A4 P08684 1/20 0.36
CYP2C9 P11712 1/20 0.36
CYP2C19 P33261 1/20 0.36
PYGL P06737 1/20 0.35
ITGB1 P05556 6/20 0.35
ITGA4 P13612 6/20 0.35
CTSA P10619 2/20 0.34
MEN1 O00255 1/20 0.34
KMT2A Q03164 1/20 0.34
HPGD P15428 1/20 0.34
P2RX7 Q99572 1/20 0.34

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL688146 0.92 CTSA (0.41) SLC22A12CYP26A1KDM4EALDH1A1CYP3A4
SCHEMBL688358 0.91 POLB (0.39) KDM4EALDH1A1CYP3A4CYP2C9CYP2C19
SCHEMBL687082 0.91 POLB (0.39) CYP26A1KDM4EALDH1A1CYP3A4CYP2C9
SCHEMBL688170 0.89 PTGER3 (0.41) SLC22A12CYP26A1KDM4EALDH1A1ITGB1
SCHEMBL687310 0.88 CTSA (0.39) KDM4EALDH1A1CYP3A4CYP2C9CYP2C19
SCHEMBL688167 0.88 SMN1; SMN2 (0.43) KDM4EALDH1A1CYP3A4CYP2C9CYP2C19
SCHEMBL693144 0.88 KDM4E (0.37) SLC22A12KDM4EALDH1A1CYP3A4CYP2C9
SCHEMBL688046 0.88 CTSA (0.42) SLC22A12CYP26A1KDM4EALDH1A1CYP3A4
SCHEMBL688149 0.88 PDE4A (0.38) SLC22A12KDM4EALDH1A1CYP3A4CYP2C9
SCHEMBL688327 0.88 SLC22A12 (0.34) SLC22A12CYP26A1KDM4EALDH1A1CYP3A4

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1203766-B1 Carboxylic acid derivatives that inhibit the binding of integrins to their receptors ENCYSIVE PHARMACEUTICALS INC (US) 2012-02-29 EP disclosed
EP-1203766-A2 Carboxylic acid derivatives that inhibit the binding of integrins to their receptors TEXAS BIOTECHNOLOGY CORPORATION (US) 2002-05-08 EP disclosed