SCHEMBL6883989

SCHEMBL6883989

Cc1nc(-c2ccc(S(C)(=O)=O)cc2)n(-c2ccc(F)cc2)n1

nearest known ligand 0.64

Predicted protein targets (top 3)

geneUniProtsupporting neighboursconfidence
PTGS2 P35354 17/20 0.64
PTGS1 P23219 4/20 0.56
AOC3 Q16853 1/20 0.51

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL5201881 1.00 PTGS2 (0.64) PTGS2PTGS1AOC3
SCHEMBL6884932 0.89 PTGS2 (0.62) PTGS2PTGS1
SCHEMBL5205568 0.88 PTGS2 (0.62) PTGS2PTGS1
SCHEMBL5203365 0.86 PTGS2 (0.57) PTGS2PTGS1
SCHEMBL6886720 0.86 PTGS2 (0.64) PTGS2PTGS1
SCHEMBL6885606 0.86 PTGS2 (0.57) PTGS2PTGS1
SCHEMBL5201916 0.86 PTGS2 (0.64) PTGS2PTGS1
SCHEMBL5207846 0.86 PTGS2 (0.62) PTGS2PTGS1
SCHEMBL6885889 0.86 PTGS2 (0.55) PTGS2PTGS1
SCHEMBL6877647 0.85 PTGS2 (0.55) PTGS2PTGS1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 5 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-6803380-B1 NON-STEROIDAL ANTIINFLAMMATORY DRUGS LABORATOIRE THERAMEX (MC) 2004-10-12 US disclosed
EP-1246809-B1 5-ARYL-1H-1,2,4-TRIAZOLE COMPOUNDS AS INHIBITORS OF CYCLOOXYGENASE-2 AND PHARMACEUTICAL COMPOSITIONS CONTAINING THEM THERAMEX (MC) 2003-07-16 EP disclosed
EP-1246809-A1 5-ARYL-1H-1,2,4-TRIAZOLE COMPOUNDS AS INHIBITORS OF CYCLOOXYGENASE-2 AND PHARMACEUTICAL COMPOSITIONS CONTAINING THEM LABORATOIRE THERAMEX (MC) 2002-10-09 EP disclosed
WO-2001034577-A1 5-ARYL-1H-1,2,4-TRIAZOLE COMPOUNDS AS INHIBITORS OF CYCLOOXYGENASE-2 AND PHARMACEUTICAL COMPOSITIONS CONTAINING THEM LABORATOIRE THERAMEX (MC) 2001-05-17 WO disclosed
EP-1099695-A1 5-aryl-1H-1,2,4-triazole compounds as inhibitors of cyclooxygenase-2 and pharmaceutical compositions containing them LABORATOIRE THERAMEX S.A. (MC) 2001-05-16 EP disclosed