SCHEMBL6885889

SCHEMBL6885889

Cc1nc(-c2ccc(S(C)(=O)=O)cc2)n(-c2ccccc2)n1

nearest known ligand 0.55

Predicted protein targets (top 4)

geneUniProtsupporting neighboursconfidence
PTGS2 P35354 14/20 0.55
ALOX5 P09917 2/20 0.53
PTGS1 P23219 2/20 0.48
SMN1; SMN2 Q16637 1/20 0.47

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL5207846 0.94 PTGS2 (0.62) PTGS2ALOX5PTGS1SMN1; SMN2
SCHEMBL6884932 0.88 PTGS2 (0.62) PTGS2ALOX5PTGS1
SCHEMBL6883989 0.86 PTGS2 (0.64) PTGS2PTGS1
SCHEMBL5201916 0.86 PTGS2 (0.64) PTGS2PTGS1
SCHEMBL6885606 0.86 PTGS2 (0.57) PTGS2ALOX5PTGS1
SCHEMBL5201881 0.86 PTGS2 (0.64) PTGS2PTGS1
SCHEMBL5203365 0.86 PTGS2 (0.57) PTGS2ALOX5PTGS1
SCHEMBL6886720 0.86 PTGS2 (0.64) PTGS2PTGS1
SCHEMBL6886482 0.85 PTGS2 (0.48) PTGS2ALOX5PTGS1
SCHEMBL7050210 0.83 PTGS2 (0.47) PTGS2ALOX5PTGS1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-6803380-B1 NON-STEROIDAL ANTIINFLAMMATORY DRUGS LABORATOIRE THERAMEX (MC) 2004-10-12 US disclosed
EP-1246809-B1 5-ARYL-1H-1,2,4-TRIAZOLE COMPOUNDS AS INHIBITORS OF CYCLOOXYGENASE-2 AND PHARMACEUTICAL COMPOSITIONS CONTAINING THEM THERAMEX (MC) 2003-07-16 EP disclosed
EP-1099695-A1 5-aryl-1H-1,2,4-triazole compounds as inhibitors of cyclooxygenase-2 and pharmaceutical compositions containing them LABORATOIRE THERAMEX S.A. (MC) 2001-05-16 EP disclosed