SCHEMBL6884237

SCHEMBL6884237

Cc1c(-c2ccc(C#N)cc2)c(C)n(Cc2ccc(C(C)(C)O)nc2)c1C

nearest known ligand 0.57

Predicted protein targets (top 10)

geneUniProtsupporting neighboursconfidence
AR P10275 9/20 0.57
CCR9 P51686 1/20 0.44
PDE10A Q9Y233 1/20 0.38
CYP11B1 P15538 3/20 0.37
KDM1A O60341 1/20 0.37
KCNH2 Q12809 1/20 0.36
CYP11B2 P19099 3/20 0.36
RET P07949 1/20 0.36
PTGDR2 Q9Y5Y4 1/20 0.35
CYP19A1 P11511 1/20 0.35

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL6464529 0.91 AR (0.69) ARCCR9PDE10ACYP11B1KDM1A
SCHEMBL6889022 0.81 AR (0.68) ARCYP11B1CYP11B2PTGDR2CYP19A1
SCHEMBL6889336 0.80 AR (0.61) ARCYP11B1KDM1ACYP11B2CYP19A1
SCHEMBL6464451 0.76 AR (0.80) ARCYP11B1KDM1ACYP11B2PTGDR2
SCHEMBL6468078 0.74 AR (0.66) ARCCR9CYP11B1KCNH2CYP11B2
SCHEMBL15147305 0.73 AR (0.58) ARCYP11B1CYP11B2PTGDR2
SCHEMBL6465291 0.73 AR (1.00) ARCYP11B1CYP11B2CYP19A1
SCHEMBL6466407 0.73 AR (0.75) ARCYP11B1CYP11B2PTGDR2CYP19A1
SCHEMBL6469502 0.73 AR (0.75) ARCYP11B1CYP11B2CYP19A1
SCHEMBL6468893 0.73 AR (0.75) ARCYP11B1CYP11B2CYP19A1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1466902-A1 ANDROGEN RECEPTOR ANTAGONISTS Takeda Chemical Industries, Ltd. (JP) 2004-10-13 EP disclosed