SCHEMBL6885382

SCHEMBL6885382

COc1ccc(-n2nc(C)nc2-c2ccc(S(C)(=O)=O)cc2)cc1OC

nearest known ligand 0.49

Predicted protein targets (top 6)

geneUniProtsupporting neighboursconfidence
CA2 P00918 6/20 0.49
CA4 P22748 6/20 0.49
CA7 P43166 6/20 0.49
CA1 P00915 3/20 0.49
PTGS2 P35354 13/20 0.47
PTGS1 P23219 2/20 0.47

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL6885799 0.86 PTGS2 (0.53) CA2CA4CA7CA1PTGS2
SCHEMBL1385685 0.84 PTGS2 (0.65) PTGS2PTGS1
SCHEMBL5205612 0.82 PTGS2 (0.61) CA2CA4CA7CA1PTGS2
SCHEMBL6884932 0.80 PTGS2 (0.62) PTGS2PTGS1
SCHEMBL6877647 0.80 PTGS2 (0.55) PTGS2PTGS1
SCHEMBL5204998 0.79 PTGS2 (0.56) PTGS2PTGS1
SCHEMBL6885817 0.79 PTGS2 (0.53) PTGS2PTGS1
SCHEMBL6883989 0.78 PTGS2 (0.64) PTGS2PTGS1
SCHEMBL5201881 0.78 PTGS2 (0.64) PTGS2PTGS1
SCHEMBL5201916 0.78 PTGS2 (0.64) PTGS2PTGS1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 5 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-6803380-B1 NON-STEROIDAL ANTIINFLAMMATORY DRUGS LABORATOIRE THERAMEX (MC) 2004-10-12 US disclosed
EP-1246809-B1 5-ARYL-1H-1,2,4-TRIAZOLE COMPOUNDS AS INHIBITORS OF CYCLOOXYGENASE-2 AND PHARMACEUTICAL COMPOSITIONS CONTAINING THEM THERAMEX (MC) 2003-07-16 EP disclosed
EP-1246809-A1 5-ARYL-1H-1,2,4-TRIAZOLE COMPOUNDS AS INHIBITORS OF CYCLOOXYGENASE-2 AND PHARMACEUTICAL COMPOSITIONS CONTAINING THEM LABORATOIRE THERAMEX (MC) 2002-10-09 EP disclosed
WO-2001034577-A1 5-ARYL-1H-1,2,4-TRIAZOLE COMPOUNDS AS INHIBITORS OF CYCLOOXYGENASE-2 AND PHARMACEUTICAL COMPOSITIONS CONTAINING THEM LABORATOIRE THERAMEX (MC) 2001-05-17 WO disclosed
EP-1099695-A1 5-aryl-1H-1,2,4-triazole compounds as inhibitors of cyclooxygenase-2 and pharmaceutical compositions containing them LABORATOIRE THERAMEX S.A. (MC) 2001-05-16 EP disclosed