SCHEMBL6887416

SCHEMBL6887416

CS(=O)(=O)CCCCC(N)=O

nearest known ligand 0.39

Predicted protein targets (top 19)

geneUniProtsupporting neighboursconfidence
KMT2A Q03164 3/20 0.39
TP53 P04637 2/20 0.39
SOAT1 P35610 2/20 0.39
ALDH1A1 P00352 2/20 0.39
LMNA P02545 2/20 0.39
MEN1 O00255 1/20 0.39
FAAH O00519 1/20 0.39
CYP1A2 P05177 1/20 0.39
CYP3A4 P08684 1/20 0.39
CYP2C19 P33261 1/20 0.39
KDM4E B2RXH2 2/20 0.35
LOX P28300 1/20 0.34
CNR1 P21554 1/20 0.32
NLRP3 Q96P20 1/20 0.32
PAOX Q6QHF9 1/20 0.31
TARDBP Q13148 1/20 0.31
PMP22 Q01453 2/20 0.30
ALOX15 P16050 1/20 0.30
BLM P54132 1/20 0.30

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL11456167 0.98 SOAT1 (0.42) KMT2ATP53SOAT1ALDH1A1LMNA
Hydrochloric Acid SCHEMBL3354872 0.98 TP53 (0.38) KMT2ATP53SOAT1ALDH1A1LMNA
SCHEMBL2810385 0.98 SOAT1 (0.42) KMT2ATP53SOAT1ALDH1A1LMNA
SCHEMBL7765920 0.98 SOAT1 (0.42) KMT2ATP53SOAT1ALDH1A1LMNA
SCHEMBL11477514 0.98 SOAT1 (0.42) KMT2ATP53SOAT1ALDH1A1LMNA
SCHEMBL6014 0.92 TP53 (0.35) KMT2ATP53SOAT1ALDH1A1LMNA
Hydrochloric Acid SCHEMBL8710297 0.90 TP53 (0.34) KMT2ATP53SOAT1ALDH1A1LMNA
SCHEMBL1161635 0.84
Hydrochloric Acid SCHEMBL5379756 0.82 NLRP3 (0.33) KMT2ATP53SOAT1ALDH1A1LMNA
SCHEMBL8629751 0.81 SPHK2 (0.48) TP53ALDH1A1LMNACYP2C19KDM4E

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 13 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
JP-2004502669-A 2004-01-29 JP claimed
EP-1353898-A2 COMPOUNDS TO TREAT ALZHEIMER'S DISEASE Elan Pharmaceuticals, Inc. (US) 2003-10-22 EP claimed
WO-2002002512-A2 COMPOUNDS TO TREAT ALZHEIMER'S DISEASE ELAN PHARMACEUTICALS, INC. (US) 2002-01-10 WO claimed
US-12371434-B2 MLL1 inhibitors and anti-cancer agents CHINA NOVARTIS INSTITUTES FOR BIOMEDICAL RESEARCH CO., LTD. (CN) 2025-07-29 US disclosed
US-20230121768-A1 MLL1 INHIBITORS AND ANTI-CANCER AGENTS CHINA NOVARTIS INSTITUTES FOR BIOMEDICAL RESEARCH CO., LTD. (CN) 2023-04-20 US disclosed
US-11407721-B2 CIS-morpholinone and other compounds as MDM2 inhibitors for the treatment of cancer AMGEN INC. (US) 2022-08-09 US disclosed
US-20180354918-A1 CIS-MORPHOLINONE AND OTHER COMPOUNDS AS MDM2 INHIBITORS FOR THE TREATMENT OF CANCER AMGEN INC. (US) 2018-12-13 US disclosed
US-20160002185-A1 CIS-MORPHOLINONE AND OTHER COMPOUNDS AS MDM2 INHIBITORS FOR THE TREATMENT OF CANCER AMGEN INC. (US) 2016-01-07 US disclosed
EP-2958902-A1 CIS-MORPHOLINONE AND OTHER COMPOUNDS AS MDM2 INHIBITORS FOR THE TREATMENT OF CANCER Amgen Inc. (US) 2015-12-30 EP disclosed
WO-2014130470-A1 CIS-MORPHOLINONE AND OTHER COMPOUNDS AS MDM2 INHIBITORS FOR THE TREATMENT OF CANCER AMGEN INC. (US) 2014-08-28 WO disclosed
EP-0765879-B1 13-Substituted milbemycin 5-oxime derivatives, their preparation and their use against insects and other pests SANKYO CO (JP) 2001-02-14 EP disclosed
US-5861429-A MITICIDES AND ANTHELMINTICS SANKYO COMPANY, LIMITED (JP) 1999-01-19 US disclosed
EP-0765879-A1 13-Substituted milbemycin 5-oxime derivatives, their preparation and their use against insects and other pests SANKYO COMPANY LIMITED (JP) 1997-04-02 EP disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (5 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-12371434-B2 MLL1 inhibitors and anti-cancer agents MLLT1, BMI1, DOT1L KMT2A 10/4885TP53 394/4885SOAT1 2512/4885
US-20180354918-A1 CIS-MORPHOLINONE AND OTHER COMPOUNDS AS MDM2 INHIBITORS FOR THE TREATMENT OF CANCER MDM2, TP53, MDM4 KMT2A 2836/4885TP53 2/4885SOAT1 3209/4885
US-11407721-B2 CIS-morpholinone and other compounds as MDM2 inhibitors for the treatment of cancer MDM2, TP53, MDM4 KMT2A 2836/4885TP53 2/4885SOAT1 3209/4885
US-20230121768-A1 MLL1 INHIBITORS AND ANTI-CANCER AGENTS MLLT1, BMI1, DOT1L KMT2A 10/4885TP53 394/4885SOAT1 2512/4885
US-20160002185-A1 CIS-MORPHOLINONE AND OTHER COMPOUNDS AS MDM2 INHIBITORS FOR THE TREATMENT OF CANCER MDM2, TP53, MDM4 KMT2A 2809/4885TP53 2/4885SOAT1 3252/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.