SCHEMBL6889863

SCHEMBL6889863

CC(C)C[C@@H](C(=O)NCC(C)(C)c1ccccc1)N(C)C(=O)OC(C)(C)C

nearest known ligand 0.53

Predicted protein targets (top 9)

geneUniProtsupporting neighboursconfidence
AAK1 Q2M2I8 4/20 0.53
MMP13 P45452 1/20 0.44
REN P00797 1/20 0.42
CTSL P07711 1/20 0.39
CTSB P07858 1/20 0.39
CTSS P25774 1/20 0.39
CTSK P43235 1/20 0.39
MMP1 P03956 1/20 0.35
L3MBTL1 Q9Y468 1/20 0.34

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL6889868 1.00 AAK1 (0.53) AAK1MMP13RENCTSLCTSB
SCHEMBL6888134 0.86 REN (0.46) AAK1MMP13RENCTSLCTSB
SCHEMBL6888131 0.86 REN (0.46) AAK1MMP13RENCTSLCTSB
SCHEMBL30807693 0.81 AAK1 (0.60) AAK1MMP13RENCTSLCTSB
SCHEMBL18414177 0.79 AAK1 (0.56) AAK1MMP13RENCTSLCTSB
SCHEMBL6892246 0.79 MAOB (0.44) MMP13REN
SCHEMBL25288616 0.78 CTSK (0.53) AAK1RENCTSLCTSBCTSS
SCHEMBL25288617 0.78 CTSK (0.53) AAK1RENCTSLCTSBCTSS
SCHEMBL29052582 0.76 CTSK (0.50) AAK1RENCTSLCTSBCTSS
SCHEMBL31512916 0.76 REN (0.59) AAK1MMP13REN

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-6737410-B1 SMOOTH MUSCLE ANTIPROLIFERATION AGENTS; SUCH AS 1-((2-(4-BENZYLOXY-PHENYL)-1-PHENETHYLCARBAMOYL-ETHYL)-METHYL-CARBAMOYL)-2 -(1H-IMIDAZOL-4-YL)-ETHYL)-CARBAMIC ACID BENZYL ESTER WARNER-LAMBERT COMPANY 2004-05-18 US disclosed
US-6265382-B1 E.G., (S--(R*, R*))-(1-((2-(4-BENZYLOXY-PHENYL)-1-PHENETHYLCARBAMOYL-ETHYL)-M ETHYL-CARBAM OYL)-2-(1H-IMIDAZOL-4-YL)-ETHYL)-CARBAMIC ACID BENZYL ESTER WARNER-LAMBERT COMPANY 2001-07-24 US disclosed