SCHEMBL689006

SCHEMBL689006

CCOC(=O)OC1=CN(C(=O)c2ccc(F)c(F)c2)CC(C)(C)c2c1n(C)c1ccccc21

nearest known ligand 0.57

Predicted protein targets (top 10)

geneUniProtsupporting neighboursconfidence
NR1H4 Q96RI1 13/20 0.57
ESR1 P03372 1/20 0.47
NR3C1 P04150 1/20 0.47
PGR P06401 1/20 0.47
NR3C2 P08235 1/20 0.47
AR P10275 1/20 0.47
PKM P14618 1/20 0.36
ELANE P08246 2/20 0.35
CNR2 P34972 2/20 0.34
MGLL Q99685 2/20 0.34

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL29880662 0.88 NR1H4 (0.70) NR1H4ESR1NR3C1PGRNR3C2
SCHEMBL273070 0.88 NR1H4 (0.70) NR1H4ESR1NR3C1PGRNR3C2
SCHEMBL4524901 0.82 NR1H4 (0.54) NR1H4ESR1NR3C1PGRNR3C2
SCHEMBL688553 0.74 NR1H4 (0.60) NR1H4ESR1NR3C1PGRNR3C2
SCHEMBL689125 0.73 NR1H4 (0.62) NR1H4ESR1NR3C1PGRNR3C2
SCHEMBL273529 0.72 NR1H4 (1.00) NR1H4ESR1NR3C1PGRNR3C2
SCHEMBL29880856 0.72 NR1H4 (1.00) NR1H4ESR1NR3C1PGRNR3C2
SCHEMBL718838 0.70 NR1H4 (0.64) NR1H4ESR1NR3C1PGRNR3C2
SCHEMBL16917651 0.69 NR1H4 (0.74) NR1H4ESR1NR3C1PGRNR3C2
SCHEMBL274281 0.69 ALDH1A1 (0.46) NR1H4PKMELANE

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1532153-B1 AZEPINOINDOLE AND PYRIDOINDOLE DERIVATIVES AS PHARMACEUTICAL AGENTS X CEPTOR THERAPEUTICS INC (US) 2012-02-29 EP claimed