SCHEMBL6890589

SCHEMBL6890589

CN(C(=O)[C@H](Cc1cn(C(c2ccccc2)(c2ccccc2)c2ccccc2)cn1)NC(=O)OCc1ccccc1)[C@@H](Cc1ccc(OCc2ccccc2)cc1)C(=O)NCC(C)(C)c1ccccc1

nearest known ligand 0.50

Predicted protein targets (top 6)

geneUniProtsupporting neighboursconfidence
HRAS P01112 2/20 0.50
SIRT2 Q8IXJ6 11/20 0.46
NMBR P28336 1/20 0.45
ITGB3 P05106 3/20 0.41
ITGA2B P08514 3/20 0.41
OPRK1 P41145 1/20 0.39

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL6890435 0.95 HRAS (0.46) HRASSIRT2NMBRITGB3ITGA2B
SCHEMBL6891485 0.90 NMBR (0.49) HRASSIRT2NMBR
SCHEMBL6890934 0.86 HRAS (0.56) HRASITGB3ITGA2B
SCHEMBL8588871 0.84 SIRT2 (0.42) HRASSIRT2NMBR
SCHEMBL6887237 0.81 HRAS (0.51) HRASITGB3ITGA2B
SCHEMBL6812617 0.79 HRAS (0.53) HRASSIRT2
SCHEMBL6812628 0.79 HRAS (0.53) HRASSIRT2
SCHEMBL6809104 0.79 HRAS (0.53) HRASSIRT2
SCHEMBL6809101 0.79 HRAS (0.53) HRASSIRT2
SCHEMBL6814437 0.77 HRAS (0.52) HRASSIRT2NMBR

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-6737410-B1 SMOOTH MUSCLE ANTIPROLIFERATION AGENTS; SUCH AS 1-((2-(4-BENZYLOXY-PHENYL)-1-PHENETHYLCARBAMOYL-ETHYL)-METHYL-CARBAMOYL)-2 -(1H-IMIDAZOL-4-YL)-ETHYL)-CARBAMIC ACID BENZYL ESTER WARNER-LAMBERT COMPANY 2004-05-18 US disclosed
US-6265382-B1 E.G., (S--(R*, R*))-(1-((2-(4-BENZYLOXY-PHENYL)-1-PHENETHYLCARBAMOYL-ETHYL)-M ETHYL-CARBAM OYL)-2-(1H-IMIDAZOL-4-YL)-ETHYL)-CARBAMIC ACID BENZYL ESTER WARNER-LAMBERT COMPANY 2001-07-24 US disclosed