SCHEMBL6890435

SCHEMBL6890435

CN(C(=O)[C@H](Cc1cn(C(c2ccccc2)(c2ccccc2)c2ccccc2)cn1)NC(=O)OCc1ccccc1)[C@@H](Cc1ccc(OCc2ccccn2)cc1)C(=O)NCC(C)(C)c1ccccc1

nearest known ligand 0.46

Predicted protein targets (top 8)

geneUniProtsupporting neighboursconfidence
HRAS P01112 1/20 0.46
SIRT2 Q8IXJ6 12/20 0.43
NMBR P28336 1/20 0.42
ITGB3 P05106 2/20 0.39
ITGA2B P08514 2/20 0.39
MAOB P27338 1/20 0.38
MEN1 O00255 1/20 0.37
KMT2A Q03164 1/20 0.37

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL6890589 0.95 HRAS (0.50) HRASSIRT2NMBRITGB3ITGA2B
SCHEMBL6887237 0.87 HRAS (0.51) HRASITGB3ITGA2BMAOBMEN1
SCHEMBL6891485 0.86 NMBR (0.49) HRASSIRT2NMBR
SCHEMBL6890934 0.81 HRAS (0.56) HRASITGB3ITGA2B
SCHEMBL6809116 0.81 HRAS (0.48) HRASSIRT2MAOB
SCHEMBL6809100 0.81 HRAS (0.48) HRASSIRT2MAOB
SCHEMBL6812563 0.80 HRAS (0.48) HRASSIRT2
SCHEMBL6812555 0.80 HRAS (0.48) HRASSIRT2
SCHEMBL8588871 0.80 SIRT2 (0.42) HRASSIRT2NMBRMAOB
SCHEMBL6892571 0.76 MAOB (0.49) HRASITGB3ITGA2BMAOB

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-6737410-B1 SMOOTH MUSCLE ANTIPROLIFERATION AGENTS; SUCH AS 1-((2-(4-BENZYLOXY-PHENYL)-1-PHENETHYLCARBAMOYL-ETHYL)-METHYL-CARBAMOYL)-2 -(1H-IMIDAZOL-4-YL)-ETHYL)-CARBAMIC ACID BENZYL ESTER WARNER-LAMBERT COMPANY 2004-05-18 US disclosed
US-6265382-B1 E.G., (S--(R*, R*))-(1-((2-(4-BENZYLOXY-PHENYL)-1-PHENETHYLCARBAMOYL-ETHYL)-M ETHYL-CARBAM OYL)-2-(1H-IMIDAZOL-4-YL)-ETHYL)-CARBAMIC ACID BENZYL ESTER WARNER-LAMBERT COMPANY 2001-07-24 US disclosed