SCHEMBL6892260

SCHEMBL6892260

COc1ccc(CCC(N)=S)cc1OC.Cc1cccc(C)c1C(N)=S

nearest known ligand 0.50

Predicted protein targets (top 12)

geneUniProtsupporting neighboursconfidence
KMT2A Q03164 3/20 0.50
MAPT P10636 2/20 0.48
KDM4E B2RXH2 1/20 0.48
ATM Q13315 1/20 0.48
CYP19A1 P11511 1/20 0.46
MEN1 O00255 2/20 0.45
CALM1 P0DP23 1/20 0.44
POLB P06746 2/20 0.44
KCNH2 Q12809 1/20 0.44
AOC3 Q16853 1/20 0.43
LMNA P02545 1/20 0.43
STAT3 P40763 1/20 0.43

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL1302702 0.86 KMT2A (0.64) KMT2AMAPTKDM4EATMCYP19A1
SCHEMBL11265688 0.74 MAPT (0.61) KMT2AMAPTKDM4EATMCYP19A1
SCHEMBL11269216 0.72 MAPT (0.64) KMT2AMAPTKDM4EATMCYP19A1
SCHEMBL28015970 0.71 ALDH1A1 (0.50) MAPTATMPOLB
SCHEMBL1032004 0.70 KDM4E (0.62) KMT2AKDM4EATMCYP19A1MEN1
SCHEMBL28176844 0.70 KDM4E (0.62) KMT2AKDM4EATMCYP19A1MEN1
SCHEMBL2403628 0.70 ATM (0.61) KMT2AMAPTKDM4EATMCYP19A1
SCHEMBL11440293 0.70 MAPT (0.60) KMT2AMAPTKDM4EATMCYP19A1
Hydrochloric Acid SCHEMBL10448977 0.69 KDM4E (0.61) KMT2AKDM4EATMCYP19A1MEN1
SCHEMBL31157848 0.69 CYP19A1 (0.77) KMT2AMAPTKDM4EATMCYP19A1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1126833-A4 OXADIAZOLE, THIADIAZOLE AND TRIAZOLE DERIVATIVES AND COMBINATORIAL LIBRARIES THEREOF TREGA BIOSCIENCES INC (US) 2004-09-08 EP claimed
EP-1126833-A2 OXADIAZOLE, THIADIAZOLE AND TRIAZOLE DERIVATIVES AND COMBINATORIAL LIBRARIES THEREOF TREGA BIOSCIENCES, INC. (US) 2001-08-29 EP claimed
WO-2000025768-A1 OXADIAZOLE, THIADIAZOLE AND TRIAZOLE DERIVATIVES AND COMBINATORIAL LIBRARIES THEREOF TREGA BIOSCIENCES, INC. (US) 2000-05-11 WO claimed