SCHEMBL6892614

SCHEMBL6892614

CC1=N[C@](Cc2cccnc2)(c2cccc(-c3cncc(Cl)c3)c2)N=C1N

nearest known ligand 0.62

Predicted protein targets (top 5)

geneUniProtsupporting neighboursconfidence
BACE1 P56817 19/20 0.62
KCNH2 Q12809 5/20 0.57
BACE2 Q9Y5Z0 2/20 0.57
APP P05067 5/20 0.45
P2RX7 Q99572 1/20 0.39

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL946753 1.00 BACE1 (0.62) BACE1KCNH2BACE2APPP2RX7
SCHEMBL6894146 0.79 BACE1 (0.56) BACE1KCNH2APP
SCHEMBL932353 0.78 BACE1 (0.69) BACE1KCNH2BACE2
SCHEMBL932732 0.77 BACE1 (1.00) BACE1KCNH2BACE2
SCHEMBL931592 0.77 BACE1 (1.00) BACE1KCNH2BACE2
SCHEMBL943862 0.76 BACE1 (0.63) BACE1KCNH2BACE2APP
SCHEMBL931789 0.76 BACE1 (0.52) BACE1KCNH2BACE2APP
SCHEMBL6891196 0.76 BACE1 (0.52) BACE1KCNH2BACE2APP
SCHEMBL6892507 0.76 BACE1 (0.52) BACE1KCNH2BACE2APP
SCHEMBL931308 0.74 BACE1 (0.63) BACE1KCNH2BACE2APP

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2011002408-A1 NOVEL COMPOUNDS FOR TREATMENT OF NEURODEGENERATION ASSOCIATED WITH DISEASES, SUCH AS ALZHEIMER'S DISEASE OR DEMENTIA ASTRAZENECA AB (SE) 2011-01-06 WO disclosed