SCHEMBL6892738

SCHEMBL6892738

CCc1ncnc(-c2ccc(C(=O)OC)cc2)c1-c1ccc(N)nc1

nearest known ligand 0.52

Predicted protein targets (top 5)

geneUniProtsupporting neighboursconfidence
PIK3CA P42336 18/20 0.52
MTOR P42345 18/20 0.52
DHFR P00374 1/20 0.43
ALOX5AP P20292 1/20 0.42
FEN1 P39748 1/20 0.42

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL6890798 0.88 PIK3CA (0.50) PIK3CAMTOR
SCHEMBL6894184 0.86 PIK3CA (0.48) PIK3CAMTORALOX5APFEN1
SCHEMBL12138100 0.85 DHFR (0.54) PIK3CAMTORDHFRALOX5APFEN1
SCHEMBL10158390 0.85 PIK3CA (0.71) PIK3CAMTOR
SCHEMBL10157564 0.84 PIK3CA (0.55) PIK3CAMTOR
SCHEMBL6892259 0.83 PIK3CA (0.57) PIK3CAMTOR
SCHEMBL6892332 0.83 PIK3CA (0.59) PIK3CAMTOR
SCHEMBL6892408 0.83 PIK3CA (0.56) PIK3CAMTOR
SCHEMBL6893262 0.83 PIK3CA (0.54) PIK3CAMTOR
SCHEMBL515738 0.82 PIK3CA (0.76) PIK3CAMTOR

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2011092198-A1 5-ALKYNYL-PYRIMIDINES BOEHRINGER INGELHEIM INTERNATIONAL GMBH (DE) 2011-08-04 WO disclosed