SCHEMBL6890798

SCHEMBL6890798

CCc1ncnc(-c2ccc(C(=O)O)cc2)c1-c1ccc(N)nc1

nearest known ligand 0.50

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
PIK3CA P42336 17/20 0.50
MTOR P42345 17/20 0.50
GABRP O00591 1/20 0.48
GABRD O14764 1/20 0.48
GABRA1 P14867 1/20 0.48
GABRB1 P18505 1/20 0.48
GABRG2 P18507 1/20 0.48
GABRB3 P28472 1/20 0.48
GABRA5 P31644 1/20 0.48
GABRA3 P34903 1/20 0.48
GABRA2 P47869 1/20 0.48
GABRB2 P47870 1/20 0.48
GABRA4 P48169 1/20 0.48
GABRE P78334 1/20 0.48
GABRA6 Q16445 1/20 0.48
GABRG1 Q8N1C3 1/20 0.48
GABRG3 Q99928 1/20 0.48
GABRQ Q9UN88 1/20 0.48
MKNK1 Q9BUB5 1/20 0.43
MKNK2 Q9HBH9 1/20 0.43

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL6892738 0.88 PIK3CA (0.52) PIK3CAMTOR
SCHEMBL6893896 0.88 PIK3CA (0.50) PIK3CAMTOR
SCHEMBL10157862 0.87 PIK3CA (0.62) PIK3CAMTOR
SCHEMBL6893410 0.86 PIK3CA (0.55) PIK3CAMTOR
SCHEMBL6893240 0.86 GABRP (0.51) PIK3CAMTORGABRPGABRDGABRA1
SCHEMBL12137685 0.85 DHFR (0.52) PIK3CAMTORGABRPGABRDGABRA1
SCHEMBL10158390 0.84 PIK3CA (0.71) PIK3CAMTOR
SCHEMBL10157307 0.84 PIK3CA (0.56) PIK3CAMTOR
SCHEMBL6892477 0.84 PIK3CA (0.50) PIK3CAMTOR
SCHEMBL6892096 0.83 PIK3CA (0.57) PIK3CAMTOR

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2011092198-A1 5-ALKYNYL-PYRIMIDINES BOEHRINGER INGELHEIM INTERNATIONAL GMBH (DE) 2011-08-04 WO disclosed