SCHEMBL6892984

SCHEMBL6892984

NCCCC(N)c1cccnc1

nearest known ligand 0.49

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
CYP2A6 P11509 1/20 0.49
HRH1 P35367 3/20 0.46
HTR2A P28223 1/20 0.46
SLC6A2 P23975 2/20 0.44
SLC6A4 P31645 2/20 0.44
SLC6A3 Q01959 2/20 0.44
CFTR P13569 1/20 0.44
GOPC Q9HD26 1/20 0.44
CHRNA7 P36544 1/20 0.43
SMN1; SMN2 Q16637 2/20 0.42
TBXAS1 P24557 1/20 0.41
KDM4E B2RXH2 1/20 0.40
GRM8 O00222 1/20 0.40
GRM4 Q14833 1/20 0.40
CYP19A1 P11511 1/20 0.40
KCNA5 P22460 3/20 0.38
ITGB3 P05106 2/20 0.38
ITGAV P06756 2/20 0.38
CYP3A4 P08684 1/20 0.38
CYP2D6 P10635 1/20 0.38

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL9189426 0.95 HRH1 (0.49) CYP2A6HRH1HTR2ASLC6A2SLC6A4
SCHEMBL30264571 0.84 SMN1; SMN2 (0.44) SLC6A2SLC6A4SLC6A3CFTRGOPC
SCHEMBL27074456 0.84 SMN1; SMN2 (0.44) SLC6A2SLC6A4SLC6A3CFTRGOPC
SCHEMBL14786230 0.84 L3MBTL1 (0.46) SLC6A2SLC6A4SLC6A3CFTRGOPC
SCHEMBL27074454 0.84 SMN1; SMN2 (0.44) SLC6A2SLC6A4SLC6A3CFTRGOPC
SCHEMBL24919476 0.82 SMN1; SMN2 (0.50) CYP2A6HRH1HTR2ASLC6A2SLC6A4
SCHEMBL28924921 0.82 SMN1; SMN2 (0.50) CYP2A6HRH1HTR2ASLC6A2SLC6A4
SCHEMBL30065165 0.82 SMN1; SMN2 (0.50) CYP2A6HRH1HTR2ASLC6A2SLC6A4
SCHEMBL28924924 0.82 SMN1; SMN2 (0.50) CYP2A6HRH1HTR2ASLC6A2SLC6A4
SCHEMBL3525890 0.81 CFTR (0.50) CYP2A6SLC6A2SLC6A4SLC6A3CFTR

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1126833-A4 OXADIAZOLE, THIADIAZOLE AND TRIAZOLE DERIVATIVES AND COMBINATORIAL LIBRARIES THEREOF TREGA BIOSCIENCES INC (US) 2004-09-08 EP claimed
EP-1126833-A2 OXADIAZOLE, THIADIAZOLE AND TRIAZOLE DERIVATIVES AND COMBINATORIAL LIBRARIES THEREOF TREGA BIOSCIENCES, INC. (US) 2001-08-29 EP claimed
WO-2000025768-A1 OXADIAZOLE, THIADIAZOLE AND TRIAZOLE DERIVATIVES AND COMBINATORIAL LIBRARIES THEREOF TREGA BIOSCIENCES, INC. (US) 2000-05-11 WO claimed