SCHEMBL6893549

SCHEMBL6893549

COc1ccc(CN2CCCc3nc(CO)sc3C2=O)cc1

nearest known ligand 0.43

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
GRM5 P41594 6/20 0.43
GAA P10253 1/20 0.43
POLB P06746 1/20 0.42
ALDH1A1 P00352 1/20 0.41
CYP1A2 P05177 1/20 0.41
CYP2C19 P33261 1/20 0.41
SMN1; SMN2 Q16637 1/20 0.41
PDE1B Q01064 1/20 0.40
HDAC3 O15379 1/20 0.39
HDAC4 P56524 1/20 0.39
HDAC1 Q13547 1/20 0.39
HDAC7 Q8WUI4 1/20 0.39
HDAC2 Q92769 1/20 0.39
HDAC10 Q969S8 1/20 0.39
HDAC11 Q96DB2 1/20 0.39
HDAC8 Q9BY41 1/20 0.39
HDAC6 Q9UBN7 1/20 0.39
HDAC9 Q9UKV0 1/20 0.39
HDAC5 Q9UQL6 1/20 0.39
LMNA P02545 2/20 0.39

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL156706 0.85 GRM5 (0.64) GRM5
SCHEMBL159565 0.76 GRM5 (0.69) GRM5
SCHEMBL1445857 0.74 GAA (0.57) GAAPOLBALDH1A1CYP1A2CYP2C19
SCHEMBL8540645 0.71 GAA (0.55) GAAPOLBALDH1A1CYP1A2CYP2C19
SCHEMBL31667380 0.71 GAA (0.43) GAAPOLBALDH1A1CYP1A2CYP2C19
SCHEMBL4509396 0.71 ACACB (0.64) GAAALDH1A1CYP1A2CYP2C19SMN1; SMN2
SCHEMBL10007682 0.70 GAA (0.48) GAAPOLBALDH1A1CYP1A2CYP2C19
SCHEMBL29135192 0.68 HDAC1 (0.51) GAAPOLBALDH1A1CYP1A2CYP2C19
SCHEMBL29135191 0.68 HDAC1 (0.51) GAAPOLBALDH1A1CYP1A2CYP2C19
SCHEMBL3459387 0.68 L3MBTL1 (0.64) GAAALDH1A1SMN1; SMN2HDAC1HDAC6

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2011073339-A1 BICYCLIC THIAZOLES AS ALLOSTERIC MODULATORS OF MGLUR5 RECEPTORS JANSSEN PHARMACEUTICA NV (BE) 2011-06-23 WO disclosed