SCHEMBL6895451

SCHEMBL6895451

Brc1ccc2[nH]c(CC3CCCCN3)nc2c1

nearest known ligand 0.47

Predicted protein targets (top 12)

geneUniProtsupporting neighboursconfidence
IDO1 P14902 4/20 0.47
POLB P06746 1/20 0.41
AAK1 Q2M2I8 1/20 0.38
HRH3 Q9Y5N1 1/20 0.38
TDO2 P48775 2/20 0.37
HTR6 P50406 2/20 0.36
CYP1A2 P05177 1/20 0.36
CYP3A4 P08684 1/20 0.36
CYP2D6 P10635 1/20 0.36
CYP2C9 P11712 1/20 0.36
CYP2C19 P33261 1/20 0.36
CACNA1H O95180 1/20 0.36

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL17516021 0.82 AAK1 (0.51) IDO1AAK1CACNA1H
SCHEMBL6896366 0.81 POLB (0.39) IDO1POLBAAK1HRH3CYP1A2
SCHEMBL12719559 0.81 IDO1 (0.53) IDO1POLBHRH3HTR6CYP1A2
SCHEMBL1255527 0.79 CACNA1H (0.43) IDO1POLBAAK1HRH3CACNA1H
Hydrochloric Acid SCHEMBL1512918 0.78 CACNA1H (0.42) IDO1POLBAAK1HRH3CACNA1H
SCHEMBL6670417 0.77 IDO1 (0.55) IDO1POLBHRH3HTR6
SCHEMBL1255702 0.77 IDO1 (0.55) IDO1POLBHRH3HTR6
SCHEMBL6893944 0.76 POLB (0.34) IDO1POLBAAK1HRH3CYP1A2
SCHEMBL1257016 0.75 CACNA1H (0.44) IDO1AAK1CYP1A2CYP3A4CYP2D6
SCHEMBL19488760 0.75 SCN10A (0.51) IDO1POLBCYP1A2CYP2D6CYP2C9

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2011031818-A2 HISTAMINE H3 INVERSE AGONISTS AND ANTAGONISTS AND METHODS OF USE THEREOF SEPRACOR INC. (US) 2011-03-17 WO disclosed
WO-2011031816-A2 HISTAMINE H3 INVERSE AGONISTS AND ANTAGONISTS AND METHODS OF USE THEREOF SEPRACOR INC. (US) 2011-03-17 WO disclosed