SCHEMBL6896366

SCHEMBL6896366

O=Cc1ccc2[nH]c(CC3CCCCN3)nc2c1

nearest known ligand 0.39

Predicted protein targets (top 13)

geneUniProtsupporting neighboursconfidence
POLB P06746 2/20 0.39
AAK1 Q2M2I8 1/20 0.36
HRH3 Q9Y5N1 1/20 0.36
CACNA1H O95180 2/20 0.34
CYP1A2 P05177 1/20 0.34
CYP3A4 P08684 1/20 0.34
CYP2D6 P10635 1/20 0.34
CYP2C9 P11712 1/20 0.34
CYP2C19 P33261 1/20 0.34
IDO1 P14902 2/20 0.34
CHEK2 O96017 1/20 0.33
KDM4E B2RXH2 2/20 0.33
CACNA1G O43497 1/20 0.33

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL6895451 0.81 IDO1 (0.47) POLBAAK1HRH3CACNA1HCYP1A2
SCHEMBL12719559 0.78 IDO1 (0.53) POLBHRH3CYP1A2CYP3A4CYP2D6
SCHEMBL1255527 0.76 CACNA1H (0.43) POLBAAK1HRH3CACNA1HIDO1
Hydrochloric Acid SCHEMBL1512918 0.75 CACNA1H (0.42) POLBAAK1HRH3CACNA1HIDO1
SCHEMBL1255702 0.74 IDO1 (0.55) POLBHRH3IDO1
SCHEMBL6670417 0.74 IDO1 (0.55) POLBHRH3IDO1
SCHEMBL6893944 0.73 POLB (0.34) POLBAAK1HRH3CACNA1HCYP1A2
SCHEMBL7649873 0.72 TDP1 (0.47) POLBKDM4E
SCHEMBL1257016 0.72 CACNA1H (0.44) AAK1CACNA1HCYP1A2CYP3A4CYP2D6
SCHEMBL1256793 0.69 POLB (0.41) POLBHRH3

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2011031816-A2 HISTAMINE H3 INVERSE AGONISTS AND ANTAGONISTS AND METHODS OF USE THEREOF SEPRACOR INC. (US) 2011-03-17 WO disclosed
WO-2011031818-A2 HISTAMINE H3 INVERSE AGONISTS AND ANTAGONISTS AND METHODS OF USE THEREOF SEPRACOR INC. (US) 2011-03-17 WO disclosed