SCHEMBL6893944

SCHEMBL6893944

CC1(C)OB(c2ccc3[nH]c(CC4CCCCN4)nc3c2)OC1(C)C

nearest known ligand 0.34

Predicted protein targets (top 15)

geneUniProtsupporting neighboursconfidence
POLB P06746 1/20 0.34
IDO1 P14902 1/20 0.33
AAK1 Q2M2I8 1/20 0.33
HRH3 Q9Y5N1 1/20 0.32
BACE1 P56817 1/20 0.31
CYP1A2 P05177 1/20 0.31
CYP3A4 P08684 1/20 0.31
CYP2D6 P10635 1/20 0.31
CYP2C9 P11712 1/20 0.31
CYP2C19 P33261 1/20 0.31
CACNA1H O95180 1/20 0.31
TLR9 Q9NR96 3/20 0.31
TLR8 Q9NR97 3/20 0.31
TLR7 Q9NYK1 3/20 0.31
HIF1A Q16665 1/20 0.31

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL13201515 0.77 DDAH1 (0.46) HIF1A
SCHEMBL6895451 0.76 IDO1 (0.47) POLBIDO1AAK1HRH3CYP1A2
SCHEMBL12567175 0.76 SCN10A (0.49) BACE1CYP1A2
SCHEMBL15746286 0.75 NPC1 (0.47) POLBCYP1A2CYP3A4CYP2D6CYP2C9
SCHEMBL28491153 0.74 NPC1 (0.35) BACE1HIF1A
SCHEMBL6896366 0.73 POLB (0.39) POLBIDO1AAK1HRH3CYP1A2
SCHEMBL12719559 0.73 IDO1 (0.53) POLBIDO1HRH3CYP1A2CYP3A4
SCHEMBL14250363 0.73 LPL (0.47) POLB
SCHEMBL18097934 0.72 LPL (0.48) POLB
SCHEMBL14327029 0.72 GAA (0.52) POLB

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2011031816-A2 HISTAMINE H3 INVERSE AGONISTS AND ANTAGONISTS AND METHODS OF USE THEREOF SEPRACOR INC. (US) 2011-03-17 WO disclosed
WO-2011031818-A2 HISTAMINE H3 INVERSE AGONISTS AND ANTAGONISTS AND METHODS OF USE THEREOF SEPRACOR INC. (US) 2011-03-17 WO disclosed