SCHEMBL6900335

SCHEMBL6900335

COc1ccc(-n2cc(O)c(=O)cc2N)cc1-c1cccc(N)c1F

nearest known ligand 0.42

Predicted protein targets (top 8)

geneUniProtsupporting neighboursconfidence
HDAC4 P56524 2/20 0.37
HDAC2 Q92769 2/20 0.37
HDAC8 Q9BY41 2/20 0.37
COMT P21964 6/20 0.35
KDM4E B2RXH2 1/20 0.34
LMNA P02545 1/20 0.34
HTR2C P28335 1/20 0.33
HTR2B P41595 1/20 0.33

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL14816318 0.87 EIF2AK3 (0.35) HDAC4HDAC2HDAC8
SCHEMBL6900956 0.77 F11 (0.39) COMTKDM4E
SCHEMBL6901682 0.72 COMT (0.55) HDAC4HDAC2HDAC8COMT
SCHEMBL6900026 0.69 COMT (0.54) HDAC4HDAC2HDAC8COMT
SCHEMBL14815910 0.68 COMT (0.39) COMT
SCHEMBL6900761 0.67 COMT (0.51) COMT
SCHEMBL6900251 0.67 SCN9A (0.40)
SCHEMBL6900936 0.67 COMT (0.48) COMT
SCHEMBL6900760 0.67 COMT (0.48) HDAC4HDAC2HDAC8COMT
SCHEMBL2468944 0.66 ROCK2 (0.36) KDM4ELMNA

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2011109254-A1 INHIBITORS OF CATECHOL O-METHYL TRANSFERASE AND THEIR USE IN THE TREATMENT OF PSYCHOTIC DISORDERS MERCK SHARP & DOHME CORP. (US) 2011-09-09 WO disclosed