SCHEMBL6901863

SCHEMBL6901863

Cc1ccc2c(ccn2C(=O)O)c1

nearest known ligand 0.55

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
TFPI2 P48307 1/20 0.55
FABP4 P15090 2/20 0.47
HTR2A P28223 1/20 0.42
HTR2C P28335 1/20 0.42
NOTUM Q6P988 1/20 0.42
OXER1 Q8TDS5 2/20 0.41
MAPT P10636 1/20 0.41
RXFP1 Q9HBX9 1/20 0.41
CYP11B1 P15538 3/20 0.40
CYP11B2 P19099 3/20 0.40
TSHR P16473 1/20 0.40
RAB9A P51151 1/20 0.40
L3MBTL1 Q9Y468 1/20 0.40
ROCK1 Q13464 1/20 0.39
THRB P10828 1/20 0.39
PIN1 Q13526 1/20 0.39
TUBB1 Q9H4B7 1/20 0.38
RAPGEF4 Q8WZA2 1/20 0.38
CYP2A6 P11509 2/20 0.38
CYP1A2 P05177 1/20 0.38

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL5622574 0.85 FABP4 (0.45) TFPI2FABP4HTR2AHTR2CNOTUM
SCHEMBL10837082 0.85 NOTUM (0.59) TFPI2FABP4HTR2AHTR2CNOTUM
SCHEMBL17782560 0.82 SNCA (0.46) TFPI2MAPTRAB9AL3MBTL1THRB
SCHEMBL5431558 0.82 RAB9A (0.66) TFPI2FABP4NOTUMMAPTTSHR
SCHEMBL4175475 0.81 TFPI2 (0.48) TFPI2FABP4HTR2AHTR2CNOTUM
SCHEMBL31517159 0.81 TFPI2 (0.48) TFPI2FABP4HTR2AHTR2CNOTUM
SCHEMBL28400587 0.81 TFPI2 (0.48) TFPI2FABP4HTR2AHTR2CNOTUM
SCHEMBL2116459 0.80 TFPI2 (0.47) TFPI2FABP4HTR2AHTR2CMAPT
SCHEMBL14220747 0.78 TFPI2 (0.62) TFPI2FABP4HTR2AHTR2CMAPT
SCHEMBL4379598 0.78 MCL1 (0.47) TFPI2FABP4HTR2AHTR2CNOTUM

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1392312-A1 TRIAZOLO 4,5-d] PYRIMIDINE DERIVATIVES AND THEIR USE AS PURINERGIC RECEPTOR ANTAGONISTS VERNALIS RESEARCH LIMITED (GB) 2004-03-03 EP disclosed
WO-2002055083-A1 TRIAZOLO[4,5-d] PYRIMIDINE DERIVATIVES AND THEIR USE AS PURINERGIC RECEPTOR ANTAGONISTS VERNALIS RESEARCH LIMITED (GB) 2002-07-18 WO disclosed