SCHEMBL6902053

SCHEMBL6902053

CCc1ccc(-c2nc[nH]n2)cc1C

nearest known ligand 0.37

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
S1PR1 P21453 6/20 0.37
S1PR3 Q99500 2/20 0.36
NOS3 P29474 1/20 0.35
NOS1 P29475 1/20 0.35
NOS2 P35228 1/20 0.35
CYP1A2 P05177 1/20 0.31
CYP2D6 P10635 1/20 0.31
CYP19A1 P11511 1/20 0.31
CYP2C9 P11712 1/20 0.31
CYP2C19 P33261 1/20 0.31
HSD17B1 P14061 1/20 0.31
ALDH1A1 P00352 2/20 0.31
KMT2A Q03164 1/20 0.31
RXRA P19793 1/20 0.31
RXRB P28702 1/20 0.31
ADH5 P11766 1/20 0.30
NOTUM Q6P988 1/20 0.30
TP53 P04637 1/20 0.30
ACACB O00763 1/20 0.30
ACACA Q13085 1/20 0.30

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL10308946 0.81 NOTUM (0.41) S1PR1S1PR3KMT2ANOTUM
SCHEMBL481728 0.77 S1PR1 (0.44) S1PR1S1PR3CYP1A2CYP2C9CYP2C19
SCHEMBL10726692 0.77 ALDH1A1 (0.53) CYP2C9CYP2C19ALDH1A1KMT2ATP53
SCHEMBL10308903 0.74 KDM4E (0.35) S1PR1S1PR3ALDH1A1KMT2ANOTUM
SCHEMBL10727144 0.74 NPC1 (0.46) ALDH1A1KMT2A
SCHEMBL4764893 0.73 NPC1 (0.35) S1PR1S1PR3
SCHEMBL16181412 0.73 NISCH (0.44) CYP2C9CYP2C19
SCHEMBL15942236 0.73 TSHR (0.43) CYP2C9CYP2C19ALDH1A1KMT2A
SCHEMBL10308948 0.73 ALDH1A1 (0.45) ALDH1A1KMT2ANOTUMTP53
SCHEMBL26110328 0.72 ADH5 (0.37) CYP19A1CYP2C9CYP2C19ALDH1A1KMT2A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2011029027-A1 SUBSTITUTED PYRAZOLO[1,5-a]PYRIMIDINE COMPOUNDS AS mTOR INHIBITORS ARRAY BIOPHARMA INC. (US) 2011-03-10 WO disclosed