SCHEMBL6902231

SCHEMBL6902231

[CH2]c1ccc(C(C)C)nc1

nearest known ligand 0.34

Predicted protein targets (top 8)

geneUniProtsupporting neighboursconfidence
CHRNA7 P36544 1/20 0.34
ESR1 P03372 2/20 0.32
ESR2 Q92731 2/20 0.32
KDM4E B2RXH2 1/20 0.31
KDM4A O75164 1/20 0.31
KDM5C P41229 1/20 0.31
KDM4D Q6B0I6 1/20 0.31
KDM4C Q9H3R0 1/20 0.31

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL9839014 0.76
SCHEMBL888893 0.75 CHRNA7 (0.36) CHRNA7ESR1ESR2KDM4EKDM4A
SCHEMBL2741630 0.73 ESR1 (0.38) CHRNA7ESR1ESR2
SCHEMBL101583 0.73 CCR1 (0.50) CHRNA7ESR1ESR2KDM4E
SCHEMBL681840 0.71 GBA1 (0.41) CHRNA7KDM4E
SCHEMBL179299 0.71 APLNR (0.51) CHRNA7ESR1ESR2
SCHEMBL18927439 0.71 CHRNA7 (0.34) CHRNA7ESR1ESR2KDM4EKDM4A
SCHEMBL21125124 0.71 TRPV4 (0.41) CHRNA7ESR1ESR2KDM4EKDM4A
SCHEMBL5371 0.71 CHRNA7 (0.44) CHRNA7ESR1ESR2KDM4E
SCHEMBL31698306 0.71 CHRNA7 (0.34) CHRNA7ESR1ESR2KDM4EKDM4A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1392312-A1 TRIAZOLO 4,5-d] PYRIMIDINE DERIVATIVES AND THEIR USE AS PURINERGIC RECEPTOR ANTAGONISTS VERNALIS RESEARCH LIMITED (GB) 2004-03-03 EP disclosed
WO-2002055083-A1 TRIAZOLO[4,5-d] PYRIMIDINE DERIVATIVES AND THEIR USE AS PURINERGIC RECEPTOR ANTAGONISTS VERNALIS RESEARCH LIMITED (GB) 2002-07-18 WO disclosed