SCHEMBL6903795

SCHEMBL6903795

CCOC(=O)c1c[nH]c2c(C3CC3)c(N3CCNCC3)c(F)cc2c1=O

nearest known ligand 0.53

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
CYP1A2 P05177 1/20 0.47
CYP3A4 P08684 1/20 0.47
CYP2C19 P33261 1/20 0.47
CLEC4M Q9H2X3 1/20 0.43
KDM4E B2RXH2 5/20 0.42
MAPT P10636 1/20 0.41
GABRA1 P14867 2/20 0.40
GABRB2 P47870 2/20 0.40
MEN1 O00255 2/20 0.39
KMT2A Q03164 2/20 0.39
GABRB1 P18505 1/20 0.39
GABRA3 P34903 1/20 0.39
ALDH1A1 P00352 3/20 0.39
HPGD P15428 3/20 0.39
HSD17B10 Q99714 3/20 0.39
BRD4 O60885 1/20 0.39
LMNA P02545 1/20 0.39
TSHR P16473 1/20 0.39
HTT P42858 1/20 0.39
CYP2J2 P51589 1/20 0.39

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL9378968 0.87 KDM4E (0.39) CYP1A2CYP3A4CYP2C19KDM4EALDH1A1
SCHEMBL1498578 0.87 PLAT (0.41) CYP1A2CYP3A4CYP2C19CLEC4MKDM4E
SCHEMBL3239412 0.85 KDM4E (0.48) CYP1A2KDM4EALDH1A1HPGDHSD17B10
Hydrochloric Acid SCHEMBL7253434 0.84 KDM4E (0.46) CYP1A2KDM4EALDH1A1HPGDHSD17B10
SCHEMBL9487698 0.83 CYP1A2 (0.56) CYP1A2CYP3A4CYP2C19CLEC4MKDM4E
SCHEMBL7517643 0.81 CYP1A2 (0.54) CYP1A2CYP3A4CYP2C19CLEC4MKDM4E
SCHEMBL5735129 0.81 KDM4E (0.39) CYP1A2KDM4EALDH1A1HPGDHSD17B10
SCHEMBL6902966 0.80 CYP1A2 (0.45) CYP1A2CYP3A4CYP2C19CLEC4MKDM4E
SCHEMBL9044874 0.79 CYP1A2 (0.43) CYP1A2CYP3A4CYP2C19CLEC4MKDM4E
SCHEMBL8898775 0.77 KDM4E (0.50) CYP2C19KDM4EMAPTMEN1KMT2A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1401829-A4 NOVEL HETEROCYCLIC ANTIBACTERIAL COMPOUNDS MICROBIOTIX INC (US) 2004-10-27 EP disclosed
EP-1401829-A1 NOVEL HETEROCYCLIC ANTIBACTERIAL COMPOUNDS Microbiotix, Inc. (US) 2004-03-31 EP disclosed
WO-2002102792-A1 NOVEL HETEROCYCLIC ANTIBACTERIAL COMPOUNDS MICROBIOTIX, INC. (US) 2002-12-27 WO disclosed