SCHEMBL6904005

SCHEMBL6904005

CCn1nc(-c2cccc(C(C)(C)N)c2)cc1Oc1ccc(-c2cnco2)cc1

nearest known ligand 0.39

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
CYP3A4 P08684 1/20 0.39
CYP2D6 P10635 1/20 0.39
LTA4H P09960 1/20 0.38
MAP4K4 O95819 1/20 0.35
MMP13 P45452 1/20 0.34
MMP14 P50281 1/20 0.34
PTGDR Q13258 1/20 0.34
CXCR1 P25024 1/20 0.34
AAK1 Q2M2I8 3/20 0.33
PORCN Q9H237 1/20 0.33
KCNH2 Q12809 1/20 0.33
HRH3 Q9Y5N1 1/20 0.33
CYP11B1 P15538 1/20 0.33
CYP11B2 P19099 1/20 0.33
MEN1 O00255 1/20 0.33
KMT2A Q03164 1/20 0.33
LMNA P02545 1/20 0.33
PKM P14618 1/20 0.33
IMPDH2 P12268 2/20 0.31
NOTUM Q6P988 1/20 0.30

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL14727791 0.85 CYP3A4 (0.35) CYP3A4CYP2D6LTA4HMMP13MMP14
SCHEMBL6902724 0.83 GPR55 (0.36) MEN1KMT2ALMNA
SCHEMBL14717787 0.83 CYP3A4 (0.33) CYP3A4CYP2D6LTA4HMMP13MMP14
SCHEMBL1659820 0.82 GPR55 (0.34) CYP3A4CXCR1
SCHEMBL1659866 0.82 GPR55 (0.39) CYP3A4CXCR1
SCHEMBL1659828 0.81 CRHR1 (0.33)
SCHEMBL1661537 0.79 GPR55 (0.32)
SCHEMBL6902469 0.73 SMN1; SMN2 (0.32) CYP3A4MEN1KMT2AGAA
SCHEMBL6904266 0.72 HRH3 (0.42) LTA4HHRH3MEN1KMT2A
SCHEMBL6902723 0.69 SCN9A (0.35) LTA4HLMNABACE1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2011046774-A1 DIARYL ETHER DERIVATIVES AS NOTCH SPARING GAMMA SECRETASE INHIBITORS MERCK SHARP & DOHME CORP. (US) 2011-04-21 WO disclosed