SCHEMBL6904049

SCHEMBL6904049

CC(C)OC(=O)N[C@@H]1CN(Cc2ccccc2)C[C@H]1c1ccc(Cl)c(F)c1

nearest known ligand 0.44

Predicted protein targets (top 13)

geneUniProtsupporting neighboursconfidence
NTRK1 P04629 10/20 0.43
DRD2 P14416 2/20 0.40
DRD4 P21917 2/20 0.40
DRD3 P35462 2/20 0.40
CHRNB2 P17787 1/20 0.39
CHRNB4 P30926 1/20 0.39
CHRNA3 P32297 1/20 0.39
CHRNA7 P36544 1/20 0.39
CHRNA4 P43681 1/20 0.39
HTR3A P46098 1/20 0.39
MAPK1 P28482 1/20 0.38
MC4R P32245 3/20 0.38
BCHE P06276 1/20 0.38

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL1975870 0.87 PDE4B (0.46) NTRK1DRD2DRD4DRD3
SCHEMBL19180711 0.87 PDE4B (0.46) NTRK1DRD2DRD4DRD3
SCHEMBL2016338 0.87 PDE4B (0.46) NTRK1DRD2DRD4DRD3
SCHEMBL16780829 0.86 NTRK1 (0.44) NTRK1DRD2DRD4DRD3MAPK1
SCHEMBL1975431 0.81 DRD2 (0.46) NTRK1DRD2DRD4DRD3
SCHEMBL2226900 0.81 DRD2 (0.46) NTRK1DRD2DRD4DRD3
SCHEMBL2413984 0.81 DPP4 (0.41) NTRK1DRD2DRD4DRD3
SCHEMBL2013229 0.79 NTRK1 (0.49) NTRK1
SCHEMBL1990123 0.79 NTRK1 (0.49) NTRK1
SCHEMBL19271023 0.79 NTRK1 (0.52) NTRK1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2011073160-A1 PYRROLIDINE DERIVATIVES AS NK - 3 RECEPTOR ANTAGONISTS F. HOFFMANN-LA ROCHE AG (CH) 2011-06-23 WO disclosed