SCHEMBL2226900

SCHEMBL2226900

COC(=O)NC1CN(Cc2ccccc2)CC1c1ccc(Cl)c(Cl)c1

nearest known ligand 0.46

Predicted protein targets (top 15)

geneUniProtsupporting neighboursconfidence
DRD2 P14416 4/20 0.46
DRD4 P21917 4/20 0.46
DRD3 P35462 4/20 0.46
SIGMAR1 Q99720 2/20 0.45
SLC6A3 Q01959 3/20 0.43
SLC6A2 P23975 1/20 0.43
SLC6A4 P31645 1/20 0.43
S1PR1 P21453 1/20 0.42
S1PR5 Q9H228 1/20 0.42
NTRK1 P04629 1/20 0.42
MEN1 O00255 1/20 0.42
KMT2A Q03164 1/20 0.42
TACR2 P21452 1/20 0.42
TACR1 P25103 1/20 0.42
RORC P51449 1/20 0.41

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL1975431 1.00 DRD2 (0.46) DRD2DRD4DRD3SIGMAR1SLC6A3
SCHEMBL1975660 0.90 PDE4B (0.48) DRD2DRD4DRD3SIGMAR1SLC6A3
SCHEMBL1984850 0.90 PDE4B (0.48) DRD2DRD4DRD3SIGMAR1SLC6A3
SCHEMBL1984852 0.90 PDE4B (0.48) DRD2DRD4DRD3SIGMAR1SLC6A3
SCHEMBL1421566 0.89 SIGMAR1 (0.47) DRD2DRD4DRD3SIGMAR1SLC6A3
SCHEMBL1421571 0.89 SIGMAR1 (0.47) DRD2DRD4DRD3SIGMAR1SLC6A3
SCHEMBL1977236 0.88 RORC (0.46) DRD2DRD4DRD3SIGMAR1RORC
SCHEMBL2225981 0.88 RORC (0.46) DRD2DRD4DRD3SIGMAR1RORC
SCHEMBL1976032 0.83 SIGMAR1 (0.47) DRD2DRD3SIGMAR1SLC6A3SLC6A2
SCHEMBL2225316 0.83 SIGMAR1 (0.47) DRD2DRD3SIGMAR1SLC6A3SLC6A2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2513052-A1 PYRROLIDINE DERIVATIVES F. Hoffmann-La Roche AG (CH) 2012-10-24 EP disclosed
WO-2011085886-A1 PYRROLIDINE DERIVATIVES F. HOFFMANN-LA ROCHE AG (CH) 2011-07-21 WO disclosed