SCHEMBL6904347

SCHEMBL6904347

CC1CN(c2cc3[nH]c(-c4ccc(F)cc4F)c(C(=O)O)c(=O)c3cc2F)CCN1

nearest known ligand 0.41

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
KDM4E B2RXH2 6/20 0.41
ALDH1A1 P00352 6/20 0.41
HPGD P15428 6/20 0.41
HSD17B10 Q99714 6/20 0.41
PMP22 Q01453 1/20 0.41
KCNH2 Q12809 2/20 0.39
PRKD3 O94806 2/20 0.39
POLB P06746 1/20 0.39
ALOX15 P16050 1/20 0.39
OPRM1 P35372 1/20 0.39
CLK2 P49760 1/20 0.39
CLK4 Q9HAZ1 1/20 0.39
TDP1 Q9NUW8 1/20 0.39
HRH3 Q9Y5N1 1/20 0.39
GSK3B P49841 2/20 0.38
PIM1 P11309 1/20 0.38
GSK3A P49840 1/20 0.38
IRAK1 P51617 1/20 0.38
RPS6KA3 P51812 1/20 0.38
DYRK1A Q13627 1/20 0.38

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL6898646 0.81 ALDH1A1 (0.44) KDM4EALDH1A1HPGDHSD17B10PMP22
(S)-Temafloxacin SCHEMBL48096 0.73 ALDH1A1 (0.61) KDM4EALDH1A1HPGDHSD17B10PMP22
Temafloxacin SCHEMBL134294 0.73 ALDH1A1 (0.61) KDM4EALDH1A1HPGDHSD17B10PMP22
Temafloxacin SCHEMBL48095 0.73 ALDH1A1 (0.61) KDM4EALDH1A1HPGDHSD17B10PMP22
Temafloxacin SCHEMBL29414891 0.73 ALDH1A1 (0.61) KDM4EALDH1A1HPGDHSD17B10PMP22
Temafloxacin SCHEMBL20769825 0.73 ALDH1A1 (0.61) KDM4EALDH1A1HPGDHSD17B10PMP22
(S)-Temafloxacin SCHEMBL9667109 0.73 ALDH1A1 (0.60) KDM4EALDH1A1HPGDHSD17B10PMP22
Temafloxacin SCHEMBL2637551 0.73 ALDH1A1 (0.62) KDM4EALDH1A1HPGDHSD17B10PMP22
Temafloxacin SCHEMBL134293 0.73 ALDH1A1 (0.62) KDM4EALDH1A1HPGDHSD17B10PMP22
Temafloxacin SCHEMBL9667105 0.73 ALDH1A1 (0.60) KDM4EALDH1A1HPGDHSD17B10PMP22

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1401829-A4 NOVEL HETEROCYCLIC ANTIBACTERIAL COMPOUNDS MICROBIOTIX INC (US) 2004-10-27 EP disclosed
EP-1401829-A1 NOVEL HETEROCYCLIC ANTIBACTERIAL COMPOUNDS Microbiotix, Inc. (US) 2004-03-31 EP disclosed
WO-2002102792-A1 NOVEL HETEROCYCLIC ANTIBACTERIAL COMPOUNDS MICROBIOTIX, INC. (US) 2002-12-27 WO disclosed