SCHEMBL6904451

SCHEMBL6904451

CCn1nc(-c2cccc(C(C)(C)NS(=O)(=O)CC(F)(F)F)c2)c(-c2ccccc2)c1Oc1ccc(C(F)(F)F)cc1

nearest known ligand 0.36

Predicted protein targets (top 18)

geneUniProtsupporting neighboursconfidence
SMN1; SMN2 Q16637 1/20 0.36
PTGDR2 Q9Y5Y4 4/20 0.36
ALDH1A1 P00352 1/20 0.34
LMNA P02545 1/20 0.34
NPSR1 Q6W5P4 1/20 0.34
RORC P51449 1/20 0.34
MAPK14 Q16539 2/20 0.33
PTGS2 P35354 4/20 0.33
NR3C1 P04150 1/20 0.32
PGR P06401 1/20 0.32
AR P10275 1/20 0.32
ESR2 Q92731 1/20 0.32
GCGR P47871 1/20 0.32
PTGS1 P23219 1/20 0.32
CETP P11597 1/20 0.32
PTGER4 P35408 1/20 0.32
SCN9A Q15858 1/20 0.31
FABP4 P15090 1/20 0.31

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL14730955 0.89 PTGDR2 (0.33) SMN1; SMN2PTGDR2RORCGCGRSCN9A
SCHEMBL1660640 0.89 PTGDR2 (0.33) SMN1; SMN2PTGDR2RORCGCGRSCN9A
SCHEMBL14717976 0.89 SMN1; SMN2 (0.33) SMN1; SMN2PTGDR2LMNARORCGCGR
SCHEMBL1660442 0.89 SMN1; SMN2 (0.33) SMN1; SMN2PTGDR2RORCGCGRSCN9A
SCHEMBL14717940 0.88 PTGDR2 (0.33) SMN1; SMN2PTGDR2RORCGCGRSCN9A
SCHEMBL14718104 0.88 PTGDR2 (0.36) SMN1; SMN2PTGDR2RORCMAPK14NR3C1
SCHEMBL14718229 0.88 POLB (0.38) SMN1; SMN2PTGDR2SCN9A
SCHEMBL14717715 0.81 PTGS2 (0.34) PTGS2SCN9A
SCHEMBL14717156 0.81 SCN9A (0.37) SCN9A
SCHEMBL14718164 0.79 LMNA (0.35) SMN1; SMN2ALDH1A1LMNANPSR1RORC

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2011046774-A1 DIARYL ETHER DERIVATIVES AS NOTCH SPARING GAMMA SECRETASE INHIBITORS MERCK SHARP & DOHME CORP. (US) 2011-04-21 WO disclosed