SCHEMBL6905689

SCHEMBL6905689

[SiH3]C(c1cccc2[nH]nnc12)(c1cccc2[nH]nnc12)c1cccc2[nH]nnc12

nearest known ligand 0.33

Predicted protein targets (top 2)

geneUniProtsupporting neighboursconfidence
AXL P30530 1/20 0.33
KIF11 P52732 1/20 0.30

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL6905674 0.87
SCHEMBL702107 0.82 KIF11 (0.42) AXLKIF11
SCHEMBL8022804 0.81 AXL (0.49) AXLKIF11
SCHEMBL1987806 0.78 GRM4 (0.33)
SCHEMBL31668752 0.77 KIF11 (0.31) AXLKIF11
SCHEMBL28473114 0.75 KIF11 (0.33) AXLKIF11
SCHEMBL30027744 0.74 KIF11 (0.36) KIF11
SCHEMBL28994959 0.74 KIF11 (0.33) KIF11
SCHEMBL15519432 0.74
SCHEMBL31619990 0.73 METAP2 (0.38) AXL

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 9 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1244517-A4 POLYMERIZATION SYSTEM WITH ORGANOSILICON COMPOUND EQUISTAR CHEM LP (US) 2004-06-30 EP disclosed
EP-1165568-A4 METAL COMPOUNDS CONTAINING NEUTRAL, MULTIDENTATE AZACYCLIC LIGANDS, CATALYSTS USING THEM, OLEFIN POLYMERIZATION METHODS USING THEM EQUISTAR CHEM LP (US) 2002-10-16 EP disclosed
EP-1244517-A1 POLYMERIZATION SYSTEM WITH ORGANOSILICON COMPOUND Equistar Chemicals L.P. (US) 2002-10-02 EP disclosed
US-6384229-B1 SILICON, TIN, GERMANIUM, OR LEAD; PYRAZOLYL, TRIAZOLYL, OR TETRAAZOLYL RING LIGAND; CATALYSTS FOR OLEFIN POLYMERIZATION EQUISTAR CHEMICALS, L.P. 2002-05-07 US disclosed
EP-1165568-A1 METAL COMPOUNDS CONTAINING NEUTRAL, MULTIDENTATE AZACYCLIC LIGANDS, CATALYSTS USING THEM, OLEFIN POLYMERIZATION METHODS USING THEM Equistar Chemicals L.P. (US) 2002-01-02 EP disclosed
WO-2001023084-A1 POLYMERIZATION SYSTEM WITH ORGANOSILICON COMPOUND EQUISTAR CHEMICALS, L.P. (US) 2001-04-05 WO disclosed
US-6180552-B1 OLEFIN POLYMERIZATION COORDINATION CATALYSTS EQUISTAR CHEMICALS, L.P. 2001-01-30 US disclosed
WO-2000059914-A1 METAL COMPOUNDS CONTAINING NEUTRAL, MULTIDENTATE AZACYCLIC LIGANDS, CATALYSTS USING THEM, OLEFIN POLYMERIZATION METHODS USING THEM EQUISTAR CHEMICALS, L.P. (US) 2000-10-12 WO disclosed
US-6093673-A USING ORGANOSILICON COMPOUND FROM PYRAZOLYL FAMILY AS EXTERNAL ADJUVANT LEADS TO INCREASED CATALYST ACTIVITY WITHOUT SACRIFICE OF STEREOREGULARITY IN POLYMERIZATION OF ALPHA OLEFINS OF THREE CARBONS OR MORE EQUISTAR CHEMICALS, LP (US) 2000-07-25 US disclosed