SCHEMBL6906119

SCHEMBL6906119

C[S+]([O-])c1ccc(-n2cc(-c3ccccc3)nc2-c2ccc(Cl)cc2)cc1

nearest known ligand 0.67

Predicted protein targets (top 9)

geneUniProtsupporting neighboursconfidence
PTGS2 P35354 11/20 0.67
PTGS1 P23219 3/20 0.48
GABRA2 P47869 2/20 0.44
GABRB2 P47870 2/20 0.44
CNR1 P21554 1/20 0.43
ALDH1A1 P00352 1/20 0.41
ALDH1A3 P47895 1/20 0.41
MAPT P10636 1/20 0.41
SMN1; SMN2 Q16637 1/20 0.41

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7059610 0.83 PTGS2 (0.64) PTGS2PTGS1GABRA2GABRB2
SCHEMBL5594726 0.81 PTGS2 (1.00) PTGS2PTGS1
SCHEMBL213892 0.81 PTGS2 (1.00) PTGS2PTGS1
SCHEMBL5594653 0.78 PTGS2 (0.78) PTGS2PTGS1
SCHEMBL5593885 0.78 PTGS2 (0.78) PTGS2PTGS1
SCHEMBL8488021 0.76 PTGS1 (0.45) PTGS2PTGS1GABRA2GABRB2ALDH1A3
SCHEMBL82549 0.75 PTGS1 (0.62) PTGS2PTGS1GABRA2GABRB2ALDH1A1
SCHEMBL21113586 0.75 PTGS2 (0.63) PTGS2PTGS1GABRA2GABRB2CNR1
SCHEMBL5698682 0.74 PTGS2 (0.90) PTGS2PTGS1
SCHEMBL3243606 0.74 PTGS2 (0.90) PTGS2PTGS1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1443942-A1 PHARMACEUTICAL COMPOSITION FOR USE FOR THE TREATMENT OF MALIGNANCIES COMPRISING IN COMBINATION A BISPHOSPHONATES, A COX-2 INHIBITOR AND A TAXOL Novartis AG (CH) 2004-08-11 EP disclosed
WO-2003035081-A1 PHARMACEUTICAL COMPOSITION FOR USE FOR THE TREATMENT OF MALIGNANCIES COMPRISING IN COMBINATION A BISPHOSPHONATES, A COX-2 INHIBITOR AND A TAXOL NOVARTIS AG (CH) 2003-05-01 WO disclosed