SCHEMBL6908693

SCHEMBL6908693

C=C(OC)C1(Cc2ccccc2)CN(Cc2ccc(Cl)cc2)CCC1=O

nearest known ligand 0.45

Predicted protein targets (top 9)

geneUniProtsupporting neighboursconfidence
NR3C1 P04150 2/20 0.45
SIGMAR1 Q99720 2/20 0.43
ALDH1A1 P00352 2/20 0.41
KDM4E B2RXH2 1/20 0.41
CYP2D6 P10635 1/20 0.40
DRD4 P21917 1/20 0.39
TACR1 P25103 1/20 0.39
CLPP Q16740 3/20 0.39
OPRL1 P41146 1/20 0.39

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL2237372 0.88 NR3C1 (0.45) NR3C1SIGMAR1ALDH1A1KDM4ECYP2D6
SCHEMBL1618300 0.82 NR3C1 (0.48) NR3C1ALDH1A1KDM4ECYP2D6TACR1
SCHEMBL21465773 0.75 CYP2D6 (0.46) NR3C1ALDH1A1KDM4ECYP2D6
SCHEMBL12487550 0.72 ABL1 (0.45) NR3C1ALDH1A1KDM4ECYP2D6
SCHEMBL5265856 0.70 CYP2D6 (0.44) NR3C1SIGMAR1ALDH1A1KDM4ECYP2D6
SCHEMBL5265862 0.70 CYP2D6 (0.44) NR3C1SIGMAR1ALDH1A1KDM4ECYP2D6
SCHEMBL15710575 0.70 KDM4E (0.50) ALDH1A1KDM4ECYP2D6
SCHEMBL3140906 0.70 KDM4E (0.46) SIGMAR1ALDH1A1KDM4EDRD4TACR1
SCHEMBL5233110 0.70 CYP2D6 (0.43) NR3C1ALDH1A1KDM4ECYP2D6TACR1
SCHEMBL5233107 0.70 CYP2D6 (0.43) NR3C1ALDH1A1KDM4ECYP2D6TACR1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2011101804-A1 PYRAZOLO PIPERIDINE DERIVATIVES AS NADPH OXIDASE INHIBITORS GENKYOTEX SA (CH) 2011-08-25 WO disclosed