Bromide

Bromide

SCHEMBL6909971

O=C(OCCNC(=O)c1cccc[n+]1CC(=O)c1ccc(Cl)cc1Cl)c1ccccc1.[Br-]

nearest known ligand 0.43

Full drug profile on Sugi Atlas →

Known targets — ChEMBL curated mechanism

ACHECHKACHRM1CHRM2CHRM3CHRM4CHRM5CHRNA1CHRNB1CHRNDCHRNECHRNGHRH2OPRM1

The experimentally established mechanism targets of Bromide. The predicted profile below is derived independently by chemical similarity — agreement is a validation signal, a miss is honest.

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
SMN1; SMN2 Q16637 3/20 0.42
KMT2A Q03164 3/20 0.39
L3MBTL1 Q9Y468 2/20 0.39
AGTR1 P30556 1/20 0.39
TMEM97 Q5BJF2 2/20 0.39
SIGMAR1 Q99720 2/20 0.39
ALDH1A1 P00352 2/20 0.39
HPGD P15428 2/20 0.39
RAB9A P51151 3/20 0.39
MITF O75030 1/20 0.39
RAD52 P43351 1/20 0.39
POLB P06746 1/20 0.38
THRB P10828 1/20 0.38
RECQL P46063 1/20 0.38
TDP1 Q9NUW8 1/20 0.38
NPC1 O15118 2/20 0.38
MAPT P10636 2/20 0.38
MAPK1 P28482 1/20 0.38
HIF1A Q16665 1/20 0.38
ERCC5 P28715 1/20 0.37

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL6908873 0.99 SMN1; SMN2 (0.43) SMN1; SMN2KMT2AL3MBTL1AGTR1TMEM97
Bromide SCHEMBL1194178 0.83 GLA (0.46) SMN1; SMN2KMT2AL3MBTL1TMEM97SIGMAR1
SCHEMBL287785 0.70 SMN1; SMN2 (0.41) SMN1; SMN2KMT2AL3MBTL1AGTR1TMEM97
Bromide SCHEMBL1194556 0.69 GLA (0.50) KMT2AL3MBTL1AGTR1ALDH1A1MITF
SCHEMBL6226750 0.69 HPGD (0.46) KMT2AL3MBTL1TMEM97SIGMAR1ALDH1A1
SCHEMBL6227326 0.68 GLA (0.48) KMT2AL3MBTL1AGTR1ALDH1A1MITF
SCHEMBL13100724 0.68 HPGD (0.74) SMN1; SMN2KMT2AALDH1A1HPGDRAB9A
Bromide SCHEMBL1194085 0.67 ALDH1A1 (0.64) SMN1; SMN2KMT2AALDH1A1HPGDRAB9A
Bromide SCHEMBL7052707 0.67 GLA (0.52) SMN1; SMN2KMT2AL3MBTL1ALDH1A1MITF
SCHEMBL6228373 0.66 ALDH1A1 (0.61) SMN1; SMN2KMT2AALDH1A1HPGDRAB9A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1222171-B1 PYRIDINIUM DERIVATIVES FOR THE MANAGEMENT OF AGING-RELATED AND DIABETIC VASCULAR COMPLICATIONS, PROCESS FOR THEIR PREPARATION AND THERAPEUTIC USES THEREOF TORRENT PHARMACEUTICALS LTD (IN) 2004-02-25 EP claimed