SCHEMBL6912585

SCHEMBL6912585

CN(C)CCc1c[nH]c2ccc(C3=CCN(C)CC3)cc12

nearest known ligand 1.00 ✓ in ChEMBL — recovers established targets

Predicted protein targets (top 8)

geneUniProtsupporting neighboursconfidence
HTR1D P28221 9/20 1.00
HTR1B P28222 9/20 1.00
HTR5A P47898 4/20 0.53
HTR1A P08908 2/20 0.51
SLC6A4 P31645 2/20 0.51
MPO P05164 1/20 0.51
HTR2A P28223 1/20 0.51
HTR2C P28335 1/20 0.51

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL29406058 1.00 HTR1D (1.00) HTR1DHTR1BHTR5AHTR1ASLC6A4
Hydrochloric Acid SCHEMBL6977751 0.99 HTR1D (0.98) HTR1DHTR1BHTR5ASLC6A4MPO
SCHEMBL6973429 0.84 HTR1D (0.73) HTR1DHTR1B
SCHEMBL6969966 0.81 HTR1D (0.67) HTR1DHTR1BHTR5AHTR1ASLC6A4
SCHEMBL6964618 0.80 HTR1D (0.66) HTR1DHTR1BHTR1A
SCHEMBL7006151 0.77 HTR1D (0.63) HTR1DHTR1BHTR5AHTR1ASLC6A4
SCHEMBL7006155 0.77 HTR1D (0.63) HTR1DHTR1BHTR5AHTR1ASLC6A4
SCHEMBL6963490 0.77 HTR1D (0.62) HTR1DHTR1BHTR5AHTR1ASLC6A4
Hydrochloric Acid SCHEMBL6977748 0.76 HTR1D (0.61) HTR1DHTR1BHTR5AHTR1ASLC6A4
SCHEMBL7008663 0.76 HTR1D (0.61) HTR1DHTR1BHTR5AHTR1ASLC6A4

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 5 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1239878-B1 FORMULATIONS OF ADENOSINE A1 AGONISTS AND 5HT1 AGONISTS GLAXO GROUP LTD (GB) 2004-02-25 EP claimed
EP-0944595-B1 5-CYCLO INDOLE COMPOUNDS AS 5-HT1D RECEPTOR LIGANDS NPS ALLELIX CORP (CA) 2003-10-01 EP claimed
US-5998438-A SEROTONIN RECEPTOR ANTAGONIST; HEADACHE THERAPY ALLELIX BIOPHARMACEUTICALS, INC. (CA) 1999-12-07 US claimed
EP-0944595-B1 5-CYCLO INDOLE COMPOUNDS AS 5-HT1D RECEPTOR LIGANDS NPS ALLELIX CORP (CA) 2003-10-01 EP disclosed
US-5998438-A SEROTONIN RECEPTOR ANTAGONIST; HEADACHE THERAPY ALLELIX BIOPHARMACEUTICALS, INC. (CA) 1999-12-07 US disclosed