SCHEMBL6918158

SCHEMBL6918158

CC(C)(C)OC(=O)N1C[C@H](O)C[C@H]1C(=O)NCc1cc(Cl)ccc1-n1cncn1

nearest known ligand 0.49

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ALDH1A1 P00352 1/20 0.49
CYP3A4 P08684 3/20 0.45
POLB P06746 2/20 0.45
CYP1A2 P05177 1/20 0.45
CYP2C19 P33261 1/20 0.45
F2 P00734 7/20 0.43
VHL P40337 1/20 0.39
MAPK8 P45983 1/20 0.37
P2RX7 Q99572 2/20 0.37
FNTA P49354 1/20 0.37
FNTB P49356 1/20 0.37
CTSL P07711 1/20 0.37
CTSB P07858 1/20 0.37
CTSS P25774 1/20 0.37
CTSK P43235 1/20 0.37
F10 P00742 1/20 0.36
F12 P00748 1/20 0.36
PRSS1 P07477 1/20 0.36
PRSS2 P07478 1/20 0.36
F7 P08709 1/20 0.36

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL6920024 0.90 ALDH1A1 (0.46) ALDH1A1CYP3A4POLBCYP1A2CYP2C19
SCHEMBL6919836 0.83 ALDH1A1 (0.55) ALDH1A1CYP3A4F2FNTAFNTB
SCHEMBL6922998 0.82 ALDH1A1 (0.43) ALDH1A1CYP3A4F2MAPK8FNTA
SCHEMBL31033414 0.80 ALDH1A1 (0.58) ALDH1A1CYP3A4POLBCYP1A2CYP2C19
SCHEMBL6077111 0.79 ALDH1A1 (0.55) ALDH1A1F2F10F12PRSS1
SCHEMBL6076941 0.79 ALDH1A1 (0.55) ALDH1A1F2F10F12PRSS1
SCHEMBL24838309 0.77 POLB (0.53) ALDH1A1CYP3A4POLBCYP1A2CYP2C19
SCHEMBL6918596 0.77 F2 (0.42) ALDH1A1CYP3A4F2F10F12
SCHEMBL6918602 0.77 F2 (0.42) ALDH1A1CYP3A4F2F10F12
SCHEMBL6921244 0.77 F2 (0.47) CYP3A4F2F10F12PRSS1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2004032834-A2 THROMBIN INHIBITORS MERCK & CO., INC. (US) 2004-04-22 WO disclosed