SCHEMBL6918296

SCHEMBL6918296

Cn1cc(-c2ccc(OCc3ccc(F)c(F)c3)c(C(=O)Nc3cccnc3)c2)cn1

nearest known ligand 0.84

Predicted protein targets (top 3)

geneUniProtsupporting neighboursconfidence
LRRK2 Q5S007 18/20 0.84
SRPK3 Q9UPE1 1/20 0.55
SGMS2 Q8NHU3 2/20 0.54

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL1647667 0.91 LRRK2 (1.00) LRRK2SRPK3SGMS2
SCHEMBL6917702 0.89 LRRK2 (0.67) LRRK2
SCHEMBL6918884 0.89 LRRK2 (1.00) LRRK2SGMS2
SCHEMBL6917994 0.88 LRRK2 (0.77) LRRK2SRPK3SGMS2
SCHEMBL6918280 0.86 LRRK2 (0.80) LRRK2SRPK3SGMS2
SCHEMBL6917228 0.86 LRRK2 (0.81) LRRK2SGMS2
SCHEMBL1647977 0.85 LRRK2 (0.80) LRRK2SGMS2
SCHEMBL6916617 0.83 LRRK2 (0.83) LRRK2SRPK3SGMS2
SCHEMBL20290865 0.82 LRRK2 (0.88) LRRK2SGMS2
SCHEMBL6917776 0.82 LRRK2 (0.78) LRRK2SGMS2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 7 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2483254-B1 NOVEL COMPOUNDS GLAXO GROUP LTD (GB) 2014-08-13 EP disclosed
EP-2483254-B1 NOVEL COMPOUNDS GLAXO GROUP LTD (GB) 2014-08-13 EP disclosed
US-8778939-B2 Compounds GLAXO GROUP LIMITED (GB) 2014-07-15 US disclosed
US-8778939-B2 Compounds GLAXO GROUP LIMITED (GB) 2014-07-15 US disclosed
US-20120184553-A1 NOVEL COMPOUNDS GLAXO GROUP LIMITED (GB) 2012-07-19 US disclosed
US-20120184553-A1 NOVEL COMPOUNDS GLAXO GROUP LIMITED (GB) 2012-07-19 US disclosed
WO-2011038572-A1 NOVEL COMPOUNDS GLAXO GROUP LIMITED (GB) 2011-04-07 WO disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (1 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20120184553-A1 NOVEL COMPOUNDS LRRK2, PARK7, PINK1 LRRK2 1/4885SRPK3 443/4885SGMS2 2320/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.