SCHEMBL6918869

SCHEMBL6918869

COc1c(Nc2cc(CNC(=O)OC(C)(C)C)c(C#N)cc2Cl)ncnc1-c1ccc(C)cc1

nearest known ligand 0.38

Predicted protein targets (top 16)

geneUniProtsupporting neighboursconfidence
AAK1 Q2M2I8 5/20 0.38
NSD2 O96028 1/20 0.37
F9 P00740 2/20 0.36
F11 P03951 1/20 0.36
F7 P08709 1/20 0.36
PRMT5 O14744 2/20 0.35
WDR77 Q9BQA1 2/20 0.35
EGFR P00533 2/20 0.34
AURKB Q96GD4 1/20 0.34
GPR119 Q8TDV5 3/20 0.34
SLC34A1 Q06495 1/20 0.33
TRPV1 Q8NER1 1/20 0.33
SRC P12931 1/20 0.33
KDR P35968 1/20 0.33
KMO O15229 1/20 0.33
TBK1 Q9UHD2 1/20 0.33

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL16300440 0.88 F9 (0.36) AAK1F9F11F7GPR119
SCHEMBL6918457 0.77 F9 (0.41) AAK1F9F11F7EGFR
SCHEMBL6920163 0.69 F9 (0.43) F9F11F7EGFRKDR
SCHEMBL30386539 0.68 PRMT5 (0.47) AAK1NSD2PRMT5WDR77
SCHEMBL9608997 0.67 TBK1 (0.45) TBK1
SCHEMBL8513739 0.67 F9 (0.44) F9F11F7EGFRSRC
SCHEMBL8509791 0.67 ROCK2 (0.44) F9F11F7SLC34A1TBK1
SCHEMBL1232774 0.66 F9 (0.53) F9F11F7SLC34A1
SCHEMBL17674434 0.66 IDO1 (0.48) AAK1NSD2PRMT5WDR77
SCHEMBL2871701 0.66 NSD2 (0.44) AAK1NSD2PRMT5WDR77

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2011017296-A1 4, 5, 6-TRISUBSTITUTED PYRIMIDINE DERIVATIVES AS FACTOR IXA INHIBITORS SCHERING CORPORATION (US) 2011-02-10 WO disclosed