SCHEMBL6919220

SCHEMBL6919220

CN1C(=O)N(Cc2ccc([S+](C)[O-])cc2)Cc2cc(C#CCn3ccnc3)ccc21

nearest known ligand 0.40

Predicted protein targets (top 9)

geneUniProtsupporting neighboursconfidence
MMP13 P45452 1/20 0.40
GPR84 Q9NQS5 1/20 0.33
CYP19A1 P11511 3/20 0.33
CYP11B1 P15538 2/20 0.33
CYP11B2 P19099 2/20 0.33
FNTA P49354 1/20 0.32
FNTB P49356 1/20 0.32
QPCT Q16769 1/20 0.31
GRM5 P41594 1/20 0.30

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL6706938 0.87 MMP13 (0.41) MMP13GPR84CYP19A1CYP11B1CYP11B2
SCHEMBL6915307 0.82 MMP13 (0.39) MMP13GRM5
SCHEMBL6917143 0.82 DRD3 (0.33) MMP13
SCHEMBL6706896 0.72 CYP3A4 (0.36) MMP13
SCHEMBL6704758 0.71 GRM5 (0.44) MMP13GRM5
SCHEMBL6706809 0.69 MMP13 (0.42) MMP13GRM5
SCHEMBL6706842 0.68 MMP13 (0.48) MMP13CYP11B1CYP11B2FNTAFNTB
SCHEMBL6706048 0.67 MMP13 (0.37) MMP13
SCHEMBL6706100 0.67 MMP13 (0.42) MMP13FNTAFNTBGRM5
SCHEMBL6706890 0.67 MMP13 (0.55) MMP13GRM5

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2004014869-A2 5,6-FUSED 3,4-DIHYDROPYRIMIDINE-2-ONE DERIVATIVES AS MATRIX METALLOPROTEINASE INHIBITORS WARNER-LAMBERT COMPANY LLC (US) 2004-02-19 WO claimed
WO-2004014869-A2 5,6-FUSED 3,4-DIHYDROPYRIMIDINE-2-ONE DERIVATIVES AS MATRIX METALLOPROTEINASE INHIBITORS WARNER-LAMBERT COMPANY LLC (US) 2004-02-19 WO disclosed