SCHEMBL6919769

SCHEMBL6919769

CC1(C)CCN[C@H]1C(=O)NC(=O)C1C[C@@H](F)CN1Cc1cc(Cl)ccc1-n1cncn1

nearest known ligand 0.36

Predicted protein targets (top 15)

geneUniProtsupporting neighboursconfidence
GPBAR1 Q8TDU6 2/20 0.36
L3MBTL1 Q9Y468 1/20 0.36
F2 P00734 4/20 0.35
NPC1 O15118 1/20 0.35
RAB9A P51151 1/20 0.35
TDP1 Q9NUW8 1/20 0.35
KMT2A Q03164 2/20 0.34
MEN1 O00255 1/20 0.34
F10 P00742 2/20 0.33
PLAT P00750 2/20 0.33
PRSS1 P07477 2/20 0.33
PRSS2 P07478 2/20 0.33
PRSS3 P35030 2/20 0.33
APOBEC3A P31941 1/20 0.33
APOBEC3G Q9HC16 1/20 0.33

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL6920701 0.85 GPBAR1 (0.38) GPBAR1L3MBTL1F2KMT2AMEN1
SCHEMBL6917424 0.84 GPBAR1 (0.38) GPBAR1L3MBTL1F2KMT2AMEN1
SCHEMBL6919210 0.82 F2 (0.39) GPBAR1L3MBTL1F2NPC1RAB9A
SCHEMBL6919199 0.82 F2 (0.39) GPBAR1L3MBTL1F2NPC1RAB9A
SCHEMBL6919773 0.81 F2 (0.40) F2F10PLATPRSS1PRSS3
SCHEMBL6922995 0.81 ALDH1A1 (0.36) GPBAR1L3MBTL1F2KMT2AMEN1
SCHEMBL6921239 0.80 F2 (0.38) GPBAR1L3MBTL1F2KMT2AMEN1
SCHEMBL6919761 0.80 F2 (0.40) GPBAR1L3MBTL1F2KMT2AMEN1
SCHEMBL6914971 0.79 MAOB (0.44) GPBAR1L3MBTL1F2KMT2AMEN1
SCHEMBL6919450 0.79 MAOB (0.44) GPBAR1L3MBTL1F2KMT2AMEN1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2004032834-A2 THROMBIN INHIBITORS MERCK & CO., INC. (US) 2004-04-22 WO claimed
WO-2004032834-A2 THROMBIN INHIBITORS MERCK & CO., INC. (US) 2004-04-22 WO disclosed