SCHEMBL6927892

SCHEMBL6927892

Clc1ccc(-c2c[nH]c(-c3ccnc(N4CCNCC4)c3)n2)cc1Cl

nearest known ligand 0.49

Predicted protein targets (top 6)

geneUniProtsupporting neighboursconfidence
DYRK1A Q13627 1/20 0.49
NMT1 P30419 16/20 0.47
PRKD3 O94806 1/20 0.46
PRKD1 Q15139 1/20 0.46
PRKD2 Q9BZL6 1/20 0.46
KARS1 Q15046 2/20 0.44

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL6927498 0.87 ITGB2 (0.41) DYRK1ANMT1
SCHEMBL6920358 0.86 CNR2 (0.52) NMT1PRKD3PRKD1
SCHEMBL6926271 0.85 TLR9 (0.45) DYRK1ANMT1
SCHEMBL6925881 0.85 PIK3C3 (0.42) DYRK1ANMT1
SCHEMBL6928153 0.83 LRRK2 (0.43) DYRK1A
SCHEMBL6923588 0.82 PIK3C3 (0.40) NMT1PRKD1
SCHEMBL6927511 0.82 WNT1 (0.41) DYRK1ANMT1PRKD1
SCHEMBL6927037 0.82 ITGB2 (0.42)
SCHEMBL6927949 0.81 ITGB2 (0.45) NMT1
SCHEMBL6925290 0.80 ITGB2 (0.41) PRKD3PRKD1PRKD2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-6514966-B2 Neuropeptide Y antagonists such as 2-chloro-5-(4-(3,4-dich loro-phenyl)-1H-imidazol-2-yl)-pyridine PFIZER INC. 2003-02-04 US disclosed
US-6355635-B1 IMIDAZOLEBENZENE, IMIDAZOLEPYRIDINE COMPOUNDS FOR TREATMENT OF OBESITY PFIZER INC. 2002-03-12 US disclosed
US-20010039277-A1 Compounds for the treatment of obesity ELLIOTT RICHARD L (US) 2001-11-08 US disclosed
WO-2000066578-A1 COMPOUNDS FOR THE TREATMENT OF OBESITY PFIZER PRODUCTS INC. (US) 2000-11-09 WO disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (1 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20010039277-A1 Compounds for the treatment of obesity NPY1R, NPY4R, NPY2R DYRK1A 1085/4885NMT1 566/4885PRKD3 1946/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.