SCHEMBL6920865

SCHEMBL6920865

COc1cccc(-c2cccc3c2nnc2c(O)n[nH]c23)c1

nearest known ligand 0.42

Predicted protein targets (top 17)

geneUniProtsupporting neighboursconfidence
SERPINE1 P05121 1/20 0.41
MAPT P10636 1/20 0.40
SMN1; SMN2 Q16637 1/20 0.40
NOTUM Q6P988 1/20 0.40
NR1H2 P55055 1/20 0.40
NR1H3 Q13133 1/20 0.40
ALDH1A1 P00352 1/20 0.40
LMNA P02545 1/20 0.40
XDH P47989 1/20 0.40
DCUN1D1 Q96GG9 1/20 0.40
PLK1 P53350 1/20 0.39
BTK Q06187 1/20 0.39
GPR84 Q9NQS5 1/20 0.39
BRD4 O60885 1/20 0.39
FYN P06241 3/20 0.39
GAA P10253 1/20 0.38
NEK1 Q96PY6 1/20 0.38

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL6919278 0.88 ENPP1 (0.43) MAPTSMN1; SMN2LMNAGAA
SCHEMBL7129327 0.85 XDH (0.42) MAPTSMN1; SMN2NOTUMNR1H2NR1H3
SCHEMBL6920075 0.85 BTK (0.48) NOTUMNR1H2NR1H3ALDH1A1LMNA
SCHEMBL6662853 0.82 CSF1R (0.50) MAPTSMN1; SMN2ALDH1A1LMNAGAA
SCHEMBL6918165 0.79 KDM4E (0.43) MAPTALDH1A1XDHDCUN1D1GAA
SCHEMBL6917745 0.77 IDO1 (0.41) MAPTSMN1; SMN2ALDH1A1LMNABTK
SCHEMBL6919881 0.75 KDM4E (0.45) ALDH1A1
SCHEMBL6918392 0.72 MAP4K4 (0.47) MAPTBTK
SCHEMBL13538503 0.71 MAPT (0.54) MAPTSMN1; SMN2NOTUMALDH1A1LMNA
SCHEMBL2662066 0.71 BTK (0.58) BTK

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2004016615-A1 PYRAZOLO (4,3c) CINNOLINE COMPOUNDS AS INHIBITORS OF ITK KINASE ACTIVITY ASTRAZENECA AB (SE) 2004-02-26 WO claimed
WO-2004016615-A1 PYRAZOLO (4,3c) CINNOLINE COMPOUNDS AS INHIBITORS OF ITK KINASE ACTIVITY ASTRAZENECA AB (SE) 2004-02-26 WO disclosed