SCHEMBL6921369

SCHEMBL6921369

C=C(Cl)c1ccc2cc(F)ccc2c1

nearest known ligand 0.46

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
CYP1A2 P05177 1/20 0.46
CYP2A6 P11509 1/20 0.46
BACE1 P56817 1/20 0.34
CES2 O00748 2/20 0.33
CES1 P23141 2/20 0.33
MAOA P21397 2/20 0.33
MAOB P27338 2/20 0.33
POLB P06746 1/20 0.33
SSTR3 P32745 1/20 0.33
HSD17B14 Q9BPX1 1/20 0.33
AHR P35869 2/20 0.32
KDM4E B2RXH2 1/20 0.32
MEN1 O00255 1/20 0.32
ALDH1A1 P00352 1/20 0.32
EGFR P00533 1/20 0.32
TP53 P04637 1/20 0.32
CYP3A4 P08684 1/20 0.32
MAPT P10636 1/20 0.32
PKM P14618 1/20 0.32
HPGD P15428 1/20 0.32

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL12520344 0.79 CYP1A2 (0.46) CYP1A2CYP2A6CES2CES1POLB
SCHEMBL7905175 0.78 CES2 (0.56) CYP1A2CYP2A6CES2CES1HSD17B14
SCHEMBL27468936 0.77 CES2 (0.48) CES2CES1MAOAMAOB
SCHEMBL22991635 0.75 CES2 (0.33) CES2CES1KDM4EMEN1ALDH1A1
SCHEMBL11722596 0.75 CYP1A2 (0.42) CYP1A2CYP2A6CES2CES1POLB
SCHEMBL27864984 0.74 CES2 (0.56) CES2CES1MEN1KMT2ASMN1; SMN2
SCHEMBL6562601 0.74 CYP1A2 (0.77) CYP1A2CYP2A6BACE1CES2CES1
SCHEMBL30366405 0.74 CYP1A2 (0.77) CYP1A2CYP2A6BACE1CES2CES1
SCHEMBL23474618 0.73 CYP2A6 (0.45) CYP1A2CYP2A6BACE1CES2CES1
SCHEMBL1769969 0.73 KDM4E (0.47) CYP1A2CYP2A6KDM4EMEN1ALDH1A1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2017192304-A1 ARYLCARBOXAMIDES AND USES THEREOF INCEPTION 1, INC. (US) 2017-11-09 WO disclosed
WO-2011061168-A1 ARYL-PYRIDINE DERIVATIVES AS ALDOSTERONE SYNTHASE INHIBITORS NOVARTIS AG (CH) 2011-05-26 WO disclosed