SCHEMBL6923488

SCHEMBL6923488

CC(CCO)CN1CCN(c2cc(-c3nc(-c4cccc(Cl)c4)c[nH]3)ccn2)CC1

nearest known ligand 0.39

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
KDM4E B2RXH2 3/20 0.39
PKM P14618 1/20 0.39
DYRK3 O43781 1/20 0.39
CCNT1 O60563 1/20 0.39
CDK9 P50750 1/20 0.39
DYRK1A Q13627 1/20 0.39
DYRK2 Q92630 1/20 0.39
DYRK1B Q9Y463 1/20 0.39
CDK1 P06493 1/20 0.38
CDK2 P24941 1/20 0.38
SMG1 Q96Q15 1/20 0.38
KMT2A Q03164 1/20 0.36
MAP3K9 P80192 1/20 0.36
MAP3K11 Q16584 1/20 0.36
ALDH1A1 P00352 2/20 0.35
MAPT P10636 2/20 0.35
LMNA P02545 1/20 0.35
HTT P42858 1/20 0.35
PIK3C3 Q8NEB9 1/20 0.35
RAD52 P43351 1/20 0.35

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL6923470 0.90 CDK1 (0.41) KDM4EPKMDYRK3CCNT1CDK9
SCHEMBL6921614 0.85 CDK1 (0.43) KDM4EPKMDYRK3CCNT1CDK9
SCHEMBL6923494 0.84 CDK1 (0.38) KDM4EPKMDYRK3CCNT1CDK9
SCHEMBL6924320 0.84 SMG1 (0.39) KDM4EPKMDYRK3CCNT1CDK9
SCHEMBL6924886 0.83 ITGB2 (0.43) KDM4EPKMDYRK3CCNT1CDK9
SCHEMBL6924959 0.82 WNT1 (0.40) DYRK1ACDK1CDK2SMG1PIK3C3
SCHEMBL6923498 0.81 CDK1 (0.39) KDM4EPKMCDK1CDK2SMG1
SCHEMBL6926669 0.81 SMG1 (0.41) KDM4EPKMDYRK3CCNT1CDK9
SCHEMBL6928029 0.81 SMG1 (0.43) KDM4EPKMDYRK3CCNT1CDK9
SCHEMBL6927962 0.81 WNT1 (0.44) KDM4EDYRK1ASMG1KMT2AALDH1A1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-6514966-B2 Neuropeptide Y antagonists such as 2-chloro-5-(4-(3,4-dich loro-phenyl)-1H-imidazol-2-yl)-pyridine PFIZER INC. 2003-02-04 US disclosed