SCHEMBL6924828

SCHEMBL6924828

Cn1c2nccc(C#N)c2c2nc(CCl)[nH]c(=O)c21

nearest known ligand 0.37

Predicted protein targets (top 9)

geneUniProtsupporting neighboursconfidence
ABCC1 P33527 1/20 0.37
DPP4 P27487 2/20 0.33
PDE5A O76074 1/20 0.31
PIM1 P11309 1/20 0.30
CDK9 P50750 1/20 0.30
GAA P10253 1/20 0.30
PARP14 Q460N5 1/20 0.30
PARP10 Q53GL7 1/20 0.30
PARP11 Q9NR21 1/20 0.30

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL6922477 0.81 GAA (0.35) DPP4PIM1GAAPARP14
SCHEMBL6924489 0.76 ABCC1 (0.41) ABCC1DPP4PIM1CDK9
SCHEMBL6924927 0.69 ABCC1 (0.48) ABCC1PIM1CDK9
SCHEMBL21072543 0.66 PARP1 (0.42) PARP14PARP10PARP11
SCHEMBL30160008 0.66 PARP1 (0.42) PARP14PARP10PARP11
SCHEMBL6923754 0.65 ABCC1 (0.43) ABCC1GAA
SCHEMBL21071874 0.63 SMN1; SMN2 (0.42) PARP14PARP10PARP11
SCHEMBL21072812 0.62 PARP14 (0.46) PARP14PARP10PARP11
SCHEMBL15549543 0.62 PDE10A (0.49)
SCHEMBL11803526 0.61 PDE5A (0.49) PDE5A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2004111052-A1 PYRROLOPYRIMIDINE DERIVATIVES AS MODULATORS OF MULTI-DRUG RESISTANCE (MDR) XENOVA LIMITED (GB) 2004-12-23 WO disclosed