SCHEMBL6924489

SCHEMBL6924489

Cn1c2nccc(C#N)c2c2nc[nH]c(=O)c21

nearest known ligand 0.41

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ABCC1 P33527 1/20 0.41
HTT P42858 1/20 0.40
IP6K1 Q92551 1/20 0.38
IP6K3 Q96PC2 1/20 0.38
IP6K2 Q9UHH9 1/20 0.38
BRD4 O60885 2/20 0.37
KDM4A O75164 4/20 0.36
KDM4B O94953 4/20 0.36
KDM5B Q9UGL1 4/20 0.36
KDM5C P41229 3/20 0.34
DPP4 P27487 1/20 0.34
PIM1 P11309 2/20 0.33
CDK9 P50750 1/20 0.33
ROCK2 O75116 3/20 0.33
ROCK1 Q13464 3/20 0.33
CDC42BPB Q9Y5S2 3/20 0.33
CDC42BPA Q5VT25 2/20 0.33
PIK3CD O00329 2/20 0.33
PIK3CA P42336 1/20 0.33
PIK3CB P42338 1/20 0.33

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL6923430 0.80 HTT (0.43) HTTIP6K1IP6K3IP6K2BRD4
SCHEMBL6924828 0.76 ABCC1 (0.37) ABCC1DPP4PIM1CDK9
SCHEMBL6924927 0.74 ABCC1 (0.48) ABCC1PIM1CDK9DYRK1A
SCHEMBL6819044 0.70 HTT (0.54) HTTIP6K1IP6K3IP6K2BRD4
SCHEMBL6822370 0.67 HTT (0.51) HTTIP6K1IP6K3IP6K2BRD4
SCHEMBL3938948 0.67 HTT (0.48) HTTBRD4ALDH1A1
SCHEMBL7127849 0.66 ADORA3 (0.47) ABCC1HTTIP6K1IP6K3IP6K2
SCHEMBL20187962 0.65 HTT (0.43) HTTIP6K1IP6K3IP6K2BRD4
SCHEMBL6920666 0.64 HTT (0.46) HTTIP6K1IP6K3IP6K2BRD4
SCHEMBL6826464 0.64 PARP1 (0.50) IP6K1BRD4KDM4AKDM4BKDM5B

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2004111052-A1 PYRROLOPYRIMIDINE DERIVATIVES AS MODULATORS OF MULTI-DRUG RESISTANCE (MDR) XENOVA LIMITED (GB) 2004-12-23 WO disclosed