SCHEMBL692526

SCHEMBL692526

CCCCCC1NCCN1

nearest known ligand 0.41

Predicted protein targets (top 12)

geneUniProtsupporting neighboursconfidence
ALDH1A1 P00352 1/20 0.41
GBA1 P04062 6/20 0.39
SPHK1 Q9NYA1 2/20 0.38
GUSB P08236 1/20 0.38
EPHX1 P07099 1/20 0.38
ALOX5 P09917 1/20 0.36
GLB1 P16278 3/20 0.36
GBA2 Q9HCG7 2/20 0.36
TSHR P16473 1/20 0.35
THRB P10828 1/20 0.35
S1PR1 P21453 1/20 0.34
S1PR3 Q99500 1/20 0.34

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL28969103 0.97 ALDH1A1 (0.44) ALDH1A1GBA1SPHK1GUSBEPHX1
SCHEMBL28815780 0.97 ALDH1A1 (0.44) ALDH1A1GBA1SPHK1GUSBEPHX1
SCHEMBL4340747 0.97 ALDH1A1 (0.44) ALDH1A1GBA1SPHK1GUSBEPHX1
SCHEMBL27992616 0.97 ALDH1A1 (0.44) ALDH1A1GBA1SPHK1GUSBEPHX1
SCHEMBL5675532 0.97 ALDH1A1 (0.44) ALDH1A1GBA1SPHK1GUSBEPHX1
SCHEMBL5675531 0.97 ALDH1A1 (0.44) ALDH1A1GBA1SPHK1GUSBEPHX1
SCHEMBL5680185 0.97 ALDH1A1 (0.44) ALDH1A1GBA1SPHK1GUSBEPHX1
SCHEMBL5677084 0.97 ALDH1A1 (0.44) ALDH1A1GBA1SPHK1GUSBEPHX1
SCHEMBL21585703 0.97 ALDH1A1 (0.44) ALDH1A1GBA1SPHK1GUSBEPHX1
SCHEMBL27992831 0.97 ALDH1A1 (0.44) ALDH1A1GBA1SPHK1GUSBEPHX1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 29 patents — showing the first 20. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0598039-B1 THERMALLY REVERSIBLE ISOCYANATE-BASED POLYMERS BATTELLE MEMORIAL INSTITUTE (US) 1998-12-09 EP claimed
EP-0848025-A2 A process for forming a finish surface on a composite material BATTELLE MEMORIAL INSTITUTE (US) 1998-06-17 EP claimed
EP-0598039-A1 THERMALLY REVERSIBLE ISOCYANATE-BASED POLYMERS BATTELLE MEMORIAL INSTITUTE (US) 1994-05-25 EP claimed
US-5239039-A Reacting an excess of hydrogen cyanide with an aryl diisocyanate; adding more diisocyanate and a dihydric phenol; crosslinking inhibition; thermally reversible; melt processible coatings and adhesives BATTELLE MEMORIAL INSTITUTE (US) 1993-08-24 US claimed
WO-1993003080-A2 THERMALLY REVERSIBLE ISOCYANATE-BASED POLYMERS BATTELLE MEMORIAL INSTITUTE (US) 1993-02-18 WO claimed
EP-0001663-A1 Novel 2-arylamino-hexahydropyrimidines and -imidazolidines, salts and complexes thereof, method of preparing the novel compounds and fungicidal compositions which contain the novel compounds DUPHAR INTERNATIONAL RESEARCH B.V (NL) 1979-05-02 EP claimed
EP-3413895-B1 C5-C6-OXACYLIC FUSED IMINOTHIADIAZINE DIOXIDE COMPOUNDS BEARING AN ETHER LINKER AS BACE INHIBITORS, COMPOSITIONS, AND THEIR USE MERCK SHARP & DOHME (US) 2021-07-21 EP disclosed
EP-2488028-B1 SUBSTITUTED PIPERIDINES THAT INCREASE P53 ACTIVITY AND THE USES THEREOF MERCK SHARP & DOHME (US) 2020-08-19 EP disclosed
EP-3223820-B1 3-METHYL-2-IMINO-HEXAHYDRO-1H-PYRANO[3,4-D]PYRIMIDIN-4-ONE COMPOUNDS AS BACE INHIBITORS, COMPOSITIONS, AND THEIR USE MERCK SHARP & DOHME (US) 2020-07-22 EP disclosed
EP-2421874-A1 COMPOSITION CONTAINING QUATERNARY AMINO-FUNCTIONAL ORGANOSILICON COMPOUNDS AND PRODUCTION AND USE THEREOF Evonik Degussa GmbH (DE) 2012-02-29 EP disclosed
WO-2010121873-A1 COMPOSITION CONTAINING QUATERNARY AMINO-FUNCTIONAL ORGANOSILICON COMPOUNDS AND PRODUCTION AND USE THEREOF EVONIK DEGUSSA GMBH (DE) 2010-10-28 WO disclosed
EP-0598039-B1 THERMALLY REVERSIBLE ISOCYANATE-BASED POLYMERS BATTELLE MEMORIAL INSTITUTE (US) 1998-12-09 EP disclosed
EP-0598039-B1 THERMALLY REVERSIBLE ISOCYANATE-BASED POLYMERS BATTELLE MEMORIAL INSTITUTE (US) 1998-12-09 EP disclosed
US-5239039-A Reacting an excess of hydrogen cyanide with an aryl diisocyanate; adding more diisocyanate and a dihydric phenol; crosslinking inhibition; thermally reversible; melt processible coatings and adhesives BATTELLE MEMORIAL INSTITUTE (US) 1993-08-24 US disclosed
WO-1993003080-A3 THERMALLY REVERSIBLE ISOCYANATE-BASED POLYMERS BATTELLE MEMORIAL INSTITUTE (US) 1993-03-18 WO disclosed
WO-1993003080-A2 THERMALLY REVERSIBLE ISOCYANATE-BASED POLYMERS BATTELLE MEMORIAL INSTITUTE (US) 1993-02-18 WO disclosed
WO-1993003080-A2 THERMALLY REVERSIBLE ISOCYANATE-BASED POLYMERS BATTELLE MEMORIAL INSTITUTE (US) 1993-02-18 WO disclosed
EP-0019906-B1 MIXTURE HARDENING UNDER THE INFLUENCE OF ATMOSPHERIC MOISTURE AND PROCESS FOR PREPARING POLYISOCYANATE POLYADDITION PRODUCTS OR CROSS-LINKED POLYEPOXIDES AKZO N.V. (NL) 1984-10-17 EP disclosed
US-4289869-A IMIDAZOLIDINE AND HEXAHYDROPYRIMIDINE DERIVATIVES AKZO NV (NL) 1981-09-15 US disclosed
EP-0019906-A1 Mixture hardening under the influence of atmospheric moisture and process for preparing polyisocyanate polyaddition products or cross-linked polyepoxides AKZO N.V. (NL) 1980-12-10 EP disclosed