SCHEMBL6925321

SCHEMBL6925321

CC(C)c1cccc(C(C)C)c1N1C(=O)c2cc3ccccc3cc2C1=O

nearest known ligand 0.66

Predicted protein targets (top 9)

geneUniProtsupporting neighboursconfidence
ANPEP P15144 8/20 0.66
DPP4 P27487 8/20 0.66
NR1H2 P55055 1/20 0.60
NR1H3 Q13133 1/20 0.60
FAAH O00519 1/20 0.41
MGLL Q99685 1/20 0.41
POLB P06746 1/20 0.38
MEN1 O00255 1/20 0.37
KMT2A Q03164 1/20 0.37

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL2820118 0.86 DPP4 (0.78) ANPEPDPP4NR1H2NR1H3FAAH
SCHEMBL29366407 0.86 DPP4 (0.78) ANPEPDPP4NR1H2NR1H3FAAH
SCHEMBL300362 0.83 DPP4 (0.61) ANPEPDPP4NR1H2NR1H3MEN1
SCHEMBL30954668 0.81 ANPEP (0.67) ANPEPDPP4NR1H2NR1H3FAAH
SCHEMBL17531021 0.81 ANPEP (0.67) ANPEPDPP4NR1H2NR1H3FAAH
SCHEMBL13171786 0.81 ANPEP (0.71) ANPEPDPP4NR1H2NR1H3
SCHEMBL173289 0.80 ANPEP (1.00) ANPEPDPP4NR1H2NR1H3
SCHEMBL9812636 0.80 ANPEP (0.69) ANPEPDPP4NR1H2NR1H3
SCHEMBL2818285 0.80 ANPEP (1.00) ANPEPDPP4NR1H2NR1H3POLB
SCHEMBL300361 0.79 DPP4 (0.60) ANPEPDPP4NR1H2NR1H3POLB

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-6515129-B1 A pharmaceutical composition which comprises, a cyclic imide derivative represented by the general formula (I): present invention relates to an aminopeptidase N inhibitor or an angiogenesis inhibitor, modulates production of tumor necrosis ISHIHARA SANGYO KAISHA LTD. (JP) 2003-02-04 US disclosed
US-6429212-B1 AMINOPEPTIDASE N INHIBITOR USED TO TREAT CANCER, TUMORS, AND RETINOPATHY; FEW SIDE EFFECTS; ANGIOGENESIS INHIBITOR ISHIHARA SANGYO KAISHA LTD. (JP) 2002-08-06 US disclosed